SCHEMBL19337459

SCHEMBL19337459

C=Nc1ccc(F)cc1/C=C\C

nearest known ligand 0.38

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
F2RL1 P55085 2/20 0.38
NFE2L2 Q16236 7/20 0.35
HRH4 Q9H3N8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18024071 0.79 KDM4E (0.36)
SCHEMBL20081417 0.79 NFE2L2 (0.34) NFE2L2
SCHEMBL20274081 0.78 ERN1 (0.32)
SCHEMBL23656272 0.78 ALDH1A1 (0.30)
SCHEMBL20274086 0.78 ERN1 (0.32)
SCHEMBL20274085 0.77 HRH4 (0.38) NFE2L2HRH4
SCHEMBL22917369 0.76 ALDH1A1 (0.34)
SCHEMBL23761786 0.76 KDM4E (0.37)
SCHEMBL9928484 0.75 MAPT (0.40)
SCHEMBL25481760 0.75 TYR (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3428162-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF BOEHRINGER INGELHEIM ANIMAL HEALTH USA INC (US) 2021-05-05 EP disclosed
EP-3428162-A1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF Merial Inc. (US) 2019-01-16 EP disclosed
EP-2922845-B1 ANTHELMINTIC COMPOUNDS AND COMPOSITIONS AND METHOD OF USING THEREOF MERIAL INC (US) 2018-06-20 EP disclosed
EP-2297133-B1 1, 2 DISUBSTITUTED HETEROCYCLIC COMPOUNDS FORUM PHARMACEUTICALS INC (US) 2017-09-13 EP disclosed