SCHEMBL19339407

SCHEMBL19339407

O=C(CBr)c1ccc2c(c1)COCc1cc(C(=O)COC(=O)[C@@H]3CCCN3)ccc1-2

nearest known ligand 0.33

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.33
ALDH1A1 P00352 4/20 0.32
TSHR P16473 1/20 0.32
MDM2 Q00987 1/20 0.32
HTT P42858 1/20 0.32
GSK3B P49841 1/20 0.32
KDM4E B2RXH2 1/20 0.32
HPGD P15428 1/20 0.32
TERT O14746 1/20 0.31
ELANE P08246 1/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
DPP4 P27487 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9977160 0.84 ALDH1A1 (0.47) ALDH1A1TSHRMDM2HTTKDM4E
SCHEMBL18213981 0.81 GSK3B (0.43) ALDH1A1TSHRMDM2GSK3BMAPT
SCHEMBL205246 0.77 PTPN1 (0.46) GSK3BMAPT
SCHEMBL15692785 0.75 MAPT (0.47) ALDH1A1TSHRMDM2GSK3BKDM4E
SCHEMBL18871030 0.75 MAPT (0.47) ALDH1A1TSHRMDM2GSK3BKDM4E
SCHEMBL18829438 0.75 L3MBTL1 (0.35) ALDH1A1TSHRMDM2HTTKDM4E
SCHEMBL203386 0.73 NPC1 (0.42) ROCK2ALDH1A1TSHRKDM4EHPGD
SCHEMBL2708423 0.73 NPC1 (0.42) ROCK2ALDH1A1TSHRKDM4EHPGD
SCHEMBL16577350 0.73 NPC1 (0.47) ALDH1A1TSHRMDM2HTTKDM4E
SCHEMBL7432130 0.72 ALDH1A1 (0.52) ALDH1A1TSHRMDM2HTTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3002281-B1 ANTIVIRAL COMPOUNDS GILEAD PHARMASSET LLC (US) 2017-09-13 EP disclosed