SCHEMBL19347372

SCHEMBL19347372

Cc1cccc(Cl)c1NC(=O)c1ccc2cccnc2c1O

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 15/20 0.59
KDR P35968 2/20 0.59
ALDH1A1 P00352 1/20 0.51
MAOB P27338 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19347295 0.92 EGLN1 (0.66) EGLN1KDRALDH1A1
SCHEMBL7684899 0.82 EGLN1 (0.63) EGLN1KDRALDH1A1
SCHEMBL7692801 0.81 KDR (0.72) EGLN1KDRALDH1A1
SCHEMBL7684545 0.81 EGLN1 (0.68) EGLN1KDRALDH1A1
SCHEMBL7691465 0.81 KDR (0.71) EGLN1KDRALDH1A1
SCHEMBL7688556 0.79 EGLN1 (0.62) EGLN1KDRALDH1A1
SCHEMBL6538253 0.79 KDR (0.67) KDR
SCHEMBL7690072 0.78 EGLN1 (0.58) EGLN1KDRALDH1A1
SCHEMBL7684517 0.78 KDR (0.61) EGLN1KDRALDH1A1
SCHEMBL6538116 0.78 ALDH1A1 (0.56) KDRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210205292-A1 INHIBITORS OF CREB-CBP INTERACTION FOR TREATMENT OF LEUKEMIA THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2021-07-08 US disclosed
WO-2017156489-A1 INHIBITORS OF CREB-CBP INTERACTION FOR TREATMENT OF LEUKEMIA THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2017-09-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210205292-A1 INHIBITORS OF CREB-CBP INTERACTION FOR TREATMENT OF LEUKEMIA CREBBP, CREB1, EP300 EGLN1 237/4885KDR 3374/4885ALDH1A1 2975/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.