SCHEMBL19360618

SCHEMBL19360618

FC(F)(F)C1CCCCN1Cc1cc2cc(Br)ccc2[nH]1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 7/20 0.39
JAK2 O60674 1/20 0.38
ROCK2 O75116 1/20 0.38
PRKD3 O94806 1/20 0.38
PRKCG P05129 1/20 0.38
PHKG2 P15735 1/20 0.38
RPS6KB1 P23443 1/20 0.38
MARK3 P27448 1/20 0.38
PRKCI P41743 1/20 0.38
CLK2 P49760 1/20 0.38
IRAK1 P51617 1/20 0.38
RPS6KA3 P51812 1/20 0.38
PRKCD Q05655 1/20 0.38
MAP4K2 Q12851 1/20 0.38
STK3 Q13188 1/20 0.38
CAMK2B Q13554 1/20 0.38
CAMK2G Q13555 1/20 0.38
CAMK2D Q13557 1/20 0.38
PKN2 Q16513 1/20 0.38
CDC42BPA Q5VT25 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19360630 0.82 HRH3 (0.51) IDO1JAK2ROCK2PRKD3PRKCG
SCHEMBL20636151 0.82 IDO1 (0.38) IDO1JAK2ROCK2PRKD3PRKCG
SCHEMBL378017 0.76 CHEK1 (0.54) IDO1CHEK1HRH3DRD2DRD3
SCHEMBL19360620 0.73 OPRM1 (0.38)
SCHEMBL19360621 0.73 HRH4 (0.52) HRH3GPR183HRH4
SCHEMBL488938 0.69 HRH3 (0.72) JAK2ROCK2PRKD3PRKCGPHKG2
SCHEMBL488937 0.69 HRH3 (0.72) JAK2ROCK2PRKD3PRKCGPHKG2
SCHEMBL28197848 0.69 GRM2 (0.41) ROCK2
SCHEMBL865591 0.65 CYP19A1 (0.50) IDO1TDO2HRH3HRH4
SCHEMBL16343090 0.64 ALDH1A1 (0.39) CHEK1DRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107531679-B Aromatic amide derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-02 CN disclosed
WO-2017157332-A1 AROMATIC AMIDE DERIVATIVE, PREPARATION METHOD THEREFOR, AND PHARMACEUTICAL APPLICATIONS THEREOF 江苏恒瑞医药股份有限公司 2017-09-21 WO disclosed