SCHEMBL19360697

SCHEMBL19360697

C=CC(=O)Nc1cccc(Nc2nc(Nc3ccc(C)cc3OC)ncc2C)c1

nearest known ligand 0.74

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
EGFR P00533 18/20 0.74
ITK Q08881 2/20 0.74
BTK Q06187 3/20 0.69
ERBB2 P04626 2/20 0.65
ERBB3 P21860 2/20 0.65
ERBB4 Q15303 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9923758 0.92 EGFR (0.82) EGFRITKBTKERBB2ERBB3
SCHEMBL9923759 0.91 EGFR (0.81) EGFRITKBTK
SCHEMBL10060098 0.89 EGFR (0.83) EGFRITKBTKERBB2ERBB3
SCHEMBL9923762 0.88 EGFR (0.82) EGFRITKBTK
SCHEMBL19360704 0.87 EGFR (0.72) EGFRITKBTK
SCHEMBL9923763 0.87 EGFR (0.82) EGFRITKBTK
SCHEMBL19360703 0.86 EGFR (0.72) EGFRITKBTKERBB4
SCHEMBL2350876 0.85 EGFR (1.00) EGFRITKBTK
SCHEMBL13606336 0.85 EGFR (1.00) EGFRITKBTK
SCHEMBL18371447 0.85 JAK3 (0.81) EGFRITKBTKERBB3ERBB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9765038-B2 Heteroaryl compounds and uses thereof CELGENE CAR LLC (BM) 2017-09-19 US disclosed