SCHEMBL19362953

SCHEMBL19362953

O=C(O)c1ccc(Oc2ccc(C3CCCCC3)cc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.53
HAO1 Q9UJM8 2/20 0.53
HDAC8 Q9BY41 2/20 0.51
HDAC6 Q9UBN7 2/20 0.51
PARP15 Q460N3 1/20 0.51
PARP10 Q53GL7 1/20 0.51
HDAC1 Q13547 1/20 0.51
SRD5A2 P31213 3/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 1/20 0.50
MAPT P10636 1/20 0.50
STAT3 P40763 3/20 0.49
KMT2A Q03164 2/20 0.49
MEN1 O00255 1/20 0.49
NPC1 O15118 1/20 0.49
POLB P06746 1/20 0.49
RAB9A P51151 1/20 0.49
BLM P54132 1/20 0.49
GPR35 Q9HC97 1/20 0.49
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21656839 1.00 KMO (0.53) KMOHAO1HDAC8HDAC6PARP15
SCHEMBL21656947 0.98 PARP10 (0.53) KMOHAO1HDAC8HDAC6PARP15
SCHEMBL21656804 0.95 PARP10 (0.53) KMOHAO1HDAC8HDAC6PARP15
SCHEMBL21274803 0.91 PARP10 (0.56) HDAC8HDAC6PARP15PARP10HDAC1
SCHEMBL31003815 0.90 KMO (0.54) KMOHAO1PARP15PARP10SRD5A2
SCHEMBL354930 0.89 KMO (0.62) KMOHAO1HDAC8HDAC6HDAC1
SCHEMBL22291720 0.89 KMO (0.62) KMOHAO1HDAC8HDAC6HDAC1
Bicarbonate SCHEMBL7018415 0.88 KMO (0.61) KMOHAO1HDAC8HDAC6HDAC1
SCHEMBL3495930 0.88 HDAC8 (0.63) KMOHAO1HDAC8HDAC6HDAC1
SCHEMBL21628450 0.85 PARP10 (0.61) HDAC8HDAC6PARP15PARP10HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3429576-B1 ENHANCERS OF NOTCH SIGNALING AND THEIR USE IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH Xeniopro GmbH (DE) 2025-10-29 EP disclosed
CN-119954697-A Aromatic molecules for the treatment of pathological conditions 赛尼欧普罗有限责任公司 2025-05-09 CN disclosed
CN-119930483-A Aromatic molecules for the treatment of pathological conditions 赛尼欧普罗有限责任公司 2025-05-06 CN disclosed
CN-118290322-A Aromatic molecules for the treatment of pathological conditions 赛尼欧普罗有限责任公司 2024-07-05 CN disclosed
US-20220354949-A1 NOVEL COMPOUNDS Xeniopro GmbH (DE) 2022-11-10 US disclosed
EP-3840834-A2 AROMATIC MOLECULES FOR USE IN THE TREATMENT OF PATHOLOGICAL CONDITIONS Xeniopro GmbH (DE) 2021-06-30 EP disclosed
CN-112888479-A Aromatic molecules for the treatment of pathological conditions 赛尼欧普罗有限责任公司 2021-06-01 CN disclosed
US-20200360355-A1 ENHANCERS OF NOTCH SIGNALING AND THEIR USE THEREOF IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH Xeniopro GmbH (DE) 2020-11-19 US disclosed
US-20200360355-A1 ENHANCERS OF NOTCH SIGNALING AND THEIR USE THEREOF IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH Xeniopro GmbH (DE) 2020-11-19 US disclosed
US-10772876-B2 Enhancers of Notch signaling and the use thereof in the treatment of cancers and malignancies medicable by upregulation of Notch Xeniopro GmbH (DE) 2020-09-15 US disclosed
US-10772876-B2 Enhancers of Notch signaling and the use thereof in the treatment of cancers and malignancies medicable by upregulation of Notch Xeniopro GmbH (DE) 2020-09-15 US disclosed
WO-2020039088-A2 NOVEL COMPOUNDS Xeniopro GmbH (DE) 2020-02-27 WO disclosed
US-20190083476-A1 ENHANCERS OF NOTCH SIGNALING AND THE USE THEREOF IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH Xeniopro GmbH (DE) 2019-03-21 US disclosed
US-20190083476-A1 ENHANCERS OF NOTCH SIGNALING AND THE USE THEREOF IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH Xeniopro GmbH (DE) 2019-03-21 US disclosed
WO-2017158190-A1 ENHANCERS OF NOTCH SIGNALING AND THEIR USE IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH Ecole polytechnique fédérale de Lausanne (EPFL) (CH) 2017-09-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220354949-A1 NOVEL COMPOUNDS MUSK, TYR, IKZF3 KMO 392/4885HAO1 2538/4885HDAC8 1020/4885
US-10772876-B2 Enhancers of Notch signaling and the use thereof in the treatment of cancers and malignancies medicable by upregulation of Notch NOTCH1, DNER, NOTCH4 KMO 2678/4885HAO1 4800/4885HDAC8 3000/4885
US-20200360355-A1 ENHANCERS OF NOTCH SIGNALING AND THEIR USE THEREOF IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH NOTCH1, DNER, NOTCH4 KMO 2754/4885HAO1 4806/4885HDAC8 2901/4885
US-20190083476-A1 ENHANCERS OF NOTCH SIGNALING AND THE USE THEREOF IN THE TREATMENT OF CANCERS AND MALIGNANCIES MEDICABLE BY UPREGULATION OF NOTCH NOTCH1, DNER, NOTCH4 KMO 2678/4885HAO1 4800/4885HDAC8 3000/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.