SCHEMBL19366305

SCHEMBL19366305

Cc1cnc(-c2cccc([C@H]3[C@H](C)[C@@H]3c3ccccc3)c2)nc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 10/20 0.64
HDAC3 O15379 2/20 0.48
HDAC7 Q8WUI4 2/20 0.48
HDAC8 Q9BY41 2/20 0.48
HDAC6 Q9UBN7 2/20 0.48
HDAC9 Q9UKV0 2/20 0.48
HDAC5 Q9UQL6 2/20 0.48
RAB9A P51151 3/20 0.38
NPC1 O15118 2/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
HPGDS O60760 4/20 0.35
ADORA1 P30542 1/20 0.35
KDR P35968 1/20 0.34
HDAC1 Q13547 1/20 0.34
NCOR2 Q9Y618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15768673 0.79 HDAC4 (1.00) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL15768960 0.77 HDAC4 (0.68) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL16602145 0.77 NPC1 (0.54) HDAC4RAB9ANPC1NFKB1NFKB2
SCHEMBL436106 0.74 NPC1 (0.65) HDAC4RAB9ANPC1NFKB1NFKB2
SCHEMBL16727393 0.73 RAB9A (0.55) HDAC4RAB9ANPC1SMN1; SMN2ADORA1
SCHEMBL29686802 0.72 MAP4K4 (0.54) HDAC4RAB9ANPC1NFKB1NFKB2
SCHEMBL17055377 0.70 NPC1 (0.67) HDAC4RAB9ANPC1NFKB1NFKB2
SCHEMBL10091200 0.70 NPC1 (0.67) HDAC4RAB9ANPC1NFKB1NFKB2
SCHEMBL15768963 0.70 HDAC4 (0.57) HDAC4HDAC3HDAC7HDAC8HDAC6
SCHEMBL15768961 0.70 HDAC4 (0.57) HDAC4HDAC3HDAC7HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9765054-B2 Histone deacetylase inhibitors and compositions and methods of use thereof CHDI FOUNDATION, INC. (US) 2017-09-19 US disclosed