SCHEMBL1940665

SCHEMBL1940665

NCCC(C(=O)O)C(=O)OCC1c2ccccc2-c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
FABP5 Q01469 3/20 0.48
FABP7 O15540 2/20 0.48
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
EPHX2 P34913 1/20 0.43
HTR2A P28223 1/20 0.42
MDM4 O15151 1/20 0.42
TP53 P04637 1/20 0.42
CASP3 P42574 2/20 0.41
CYP1A2 P05177 1/20 0.40
TSHR P16473 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14947096 1.00 KMT2A (0.52) KMT2AFABP5FABP7CA1CA2
SCHEMBL97613 0.92 KMT2A (0.50) KMT2AFABP5FABP7CA1CA2
SCHEMBL25144 0.91 KMT2A (0.49) KMT2AFABP5FABP7CA1CA2
SCHEMBL3976225 0.89 KMT2A (0.48) KMT2AFABP5FABP7CA1CA2
SCHEMBL525558 0.89 KMT2A (0.48) KMT2AFABP5FABP7CA1CA2
SCHEMBL524545 0.89 KMT2A (0.48) KMT2AFABP5FABP7CA1CA2
SCHEMBL3426738 0.89 KMT2A (0.48) KMT2AFABP5FABP7CA1CA2
SCHEMBL28036073 0.89 KMT2A (0.48) KMT2AFABP5FABP7CA1CA2
SCHEMBL524835 0.89 KMT2A (0.48) KMT2AFABP5FABP7CA1CA2
SCHEMBL1162471 0.88 KMT2A (0.55) KMT2AFABP5FABP7CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 88 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3455234-B1 SECO MACROLIDE COMPOUNDS SELVITA D O O (HR) 2026-04-01 EP disclosed
WO-2025224092-A1 PEPTIDE-BASED RADIOPHARMACEUTICALS FOR NON-INVASIVE IMAGING OF THE FUNCTIONAL LIVER RESERVE MEDIZINISCHE UNIVERSITÄT INNSBRUCK (AT) 2025-10-30 WO disclosed
EP-4640240-A1 PEPTIDE-BASED RADIOPHARMACEUTICALS FOR NON-INVASIVE IMAGING OF THE FUNCTIONAL LIVER RESERVE Medizinische Universität Innsbruck (AT) 2025-10-29 EP disclosed
US-20250129125-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF GENENTECH, INC. (US) 2025-04-24 US disclosed
US-12187816-B2 Macrocyclic compounds and methods of use thereof GENENTECH, INC. (US) 2025-01-07 US disclosed
US-20240218021-A1 CYCLIN INHIBITORS CIRCLE PHARMA, INC. 2024-07-04 US disclosed
US-12023378-B2 Covalently linked antigen-antibody conjugates HOFFMANN-LA ROCHE INC. (US) 2024-07-02 US disclosed
CN-118085061-A Cyclic peptide tyrosine compounds as neuropeptide y receptor modulators 詹森药业有限公司 2024-05-28 CN disclosed
CN-110099692-B Cyclic peptide tyrosine compounds as neuropeptide y receptor modulators 詹森药业有限公司 2024-03-12 CN disclosed
CN-117295525-A Cell penetrating peptide conjugates and methods of use thereof 牛津大学科技创新有限公司 2023-12-26 CN disclosed
US-5854410-A Oligonucleoside cleavage compounds and therapies GENTA INCORPORATED (US) 1998-12-29 US disclosed
EP-0542887-B1 PSORALEN CONJUGATED METHYLPHOSPHONATE OLIGONUCLEOTIDES AS THERAPEUTIC AGENTS FOR CHRONIC MYELOGENOUS LEUKEMIA GENTA INC (US) 1998-12-02 EP disclosed
EP-0542928-A4 IMPROVED NON-NUCLEOTIDE-BASED LINKER REAGENTS FOR OLIGOMERS GENTA INC (US) 1994-07-27 EP disclosed
EP-0542928-A1 IMPROVED NON-NUCLEOTIDE-BASED LINKER REAGENTS FOR OLIGOMERS GENTA INCORPORATED (US) 1993-05-26 EP disclosed
EP-0542887-A1 PSORALEN CONJUGATED METHYLPHOSPHONATE OLIGONUCLEOTIDES AS THERAPEUTIC AGENTS FOR CHRONIC MYELOGENOUS LEUKEMIA GENTA INCORPORATED (US) 1993-05-26 EP disclosed
EP-0541663-A1 PEPTIDES AND PHARMACEUTICAL COMPOSITIONS HAVING GLYCOPROTEIN HORMONE AGONISTIC OR ANTAGONISTIC ACTIVITY STICHTING CENTRAAL DIERGENEESKUNDIG INSTITUUT (NL) 1993-05-19 EP disclosed
WO-1992002542-A1 PEPTIDES AND PHARMACEUTICAL COMPOSITIONS HAVING GLYCOPROTEIN HORMONE AGONISTIC OR ANTAGONISTIC ACTIVITY STICHTING CENTRAAL DIERGENEESKUNDIG INSTITUUT (NL) 1992-02-20 WO disclosed
WO-1992002641-A1 PSORALEN CONJUGATED METHYLPHOSPHONATE OLIGONUCLEOTIDES AS THERAPEUTIC AGENTS FOR CHRONIC MYELOGENOUS LEUKEMIA GENTA INCORPORATED (US) 1992-02-20 WO disclosed
WO-1992002532-A1 IMPROVED NON-NUCLEOTIDE-BASED LINKER REAGENTS FOR OLIGOMERS GENTA INCORPORATED (US) 1992-02-20 WO disclosed
EP-0339695-A2 A process for preparing an antigenic or immunogenic conjugate as well as the use of such conjugates STICHTING VOOR DE TECHNISCHE WETENSCHAPPEN (NL) 1989-11-02 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12187816-B2 Macrocyclic compounds and methods of use thereof PAICS, CYCS, LSS KMT2A 2834/4885FABP5 4000/4885FABP7 2688/4885
US-20250129125-A1 MACROCYCLIC COMPOUNDS AND METHODS OF USE THEREOF PAICS, CYCS, LSS KMT2A 2834/4885FABP5 4000/4885FABP7 2688/4885
US-20240218021-A1 CYCLIN INHIBITORS CCNI, CCNC, CDK2 KMT2A 1479/4885FABP5 3119/4885FABP7 3683/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.