SCHEMBL19409889

SCHEMBL19409889

CCCCC(=O)N=C(N)N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.46
CES2 O00748 5/20 0.46
LMNA P02545 1/20 0.45
ALDH1A1 P00352 3/20 0.42
TP53 P04637 2/20 0.42
CA1 P00915 1/20 0.41
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
FAAH O00519 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38
SOAT1 P35610 1/20 0.38
AKR1B1 P15121 1/20 0.37
DDAH1 O94760 1/20 0.37
BACE1 P56817 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
TSHR P16473 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28419426 0.93 CES2 (0.48) CES1CES2ALDH1A1TP53MEN1
SCHEMBL11296708 0.91 CES2 (0.50) CES1CES2ALDH1A1TP53MEN1
SCHEMBL11025699 0.91 CES2 (0.50) CES1CES2ALDH1A1TP53MEN1
SCHEMBL11288198 0.91 CES2 (0.50) CES1CES2ALDH1A1TP53MEN1
Hydrochloric Acid SCHEMBL28349226 0.91 CES2 (0.46) CES1CES2ALDH1A1TP53MEN1
SCHEMBL11294421 0.91 CES2 (0.50) CES1CES2ALDH1A1TP53MEN1
SCHEMBL10734667 0.85
SCHEMBL21351040 0.81 FAAH (0.68) LMNATP53MEN1KMT2AFAAH
SCHEMBL19661878 0.81 FAAH (0.62) LMNATP53MEN1KMT2AFAAH
SCHEMBL15474220 0.78 CES1 (0.48) CES1CES2ALDH1A1TP53CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10744179-B2 Method for treatment of inflammatory skin disorders with inhibitors of IL-36 proteolytic processing The Provost, Fellows, Foundation Scholars, & the Other Members of Board, of The College of the Holy (IE) 2020-08-18 US disclosed
US-20170281716-A1 USE OF INHIBITORS OF IL-36 PROTEOLYTIC PROCESSING FOR THE TREATMENT AND/OR REDUCTION OF INFLAMMATION The Provost, Fellows, Foundation Scholars, & the Other Members of Board, of The College of the Holy (IE) 2017-10-05 US disclosed
CN-1107836-A Novel substituted guanidine derivatives, their preparation and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-09-06 CN disclosed
CN-1028592-C Insecticidal composition containing novel substituted guanidine derivative and application TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-05-31 CN disclosed
CN-1059719-A Novel substituted guanidine derivatives, their preparation and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1992-03-25 CN disclosed