SCHEMBL19418484

SCHEMBL19418484

Fc1ccc(NCC2CC2)nc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRHR1 P34998 4/20 0.54
ABL1 P00519 1/20 0.49
AOC3 Q16853 1/20 0.44
PDE10A Q9Y233 1/20 0.41
TRPA1 O75762 1/20 0.41
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GABRA5 P31644 1/20 0.41
FLT3 P36888 1/20 0.40
TYRO3 Q06418 1/20 0.40
MERTK Q12866 1/20 0.40
GAS6 Q14393 1/20 0.40
GPR39 O43194 1/20 0.40
KCNH2 Q12809 1/20 0.40
CYP2D6 P10635 1/20 0.39
DPP4 P27487 1/20 0.39
DPP8 Q6V1X1 1/20 0.39
DPP9 Q86TI2 1/20 0.39
DPP7 Q9UHL4 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21920755 0.79 CRHR1 (0.48) CRHR1PDE10AKDM4ETSHRHSD17B10
SCHEMBL17141620 0.79 NPC1 (0.48) PDE10AKDM4ETSHRHSD17B10GPR39
SCHEMBL13685171 0.79 PDE10A (0.41) CRHR1ABL1PDE10AKDM4ETSHR
SCHEMBL1108661 0.79 CRHR1 (0.51) CRHR1ABL1PDE10AKDM4ETSHR
SCHEMBL4037459 0.79 PDE10A (0.41) CRHR1ABL1PDE10AKDM4ETSHR
SCHEMBL17141822 0.79 PDE10A (0.44) CRHR1PDE10AKDM4ETSHRHSD17B10
SCHEMBL16030699 0.77 USP30 (0.42) CRHR1KDM4ETSHRHSD17B10CYP2D6
SCHEMBL16030698 0.77 USP30 (0.42) CRHR1KDM4ETSHRHSD17B10CYP2D6
SCHEMBL30775294 0.76 KCNH2 (0.48) ABL1FLT3TYRO3MERTKGAS6
SCHEMBL4033485 0.75 GPR39 (0.40) CRHR1ABL1PDE10AKDM4ETSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2925757-B1 COMPOUNDS AND COMPOSITIONS FOR THE TREATMENT OF PARASITIC DISEASES NOVARTIS AG (CH) 2017-10-04 EP disclosed