SCHEMBL19446089

SCHEMBL19446089

CCc1cnc(OC(C)C)c(OC)c1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 2/20 0.43
DHODH Q02127 1/20 0.39
TRPM8 Q7Z2W7 1/20 0.38
HTR2A P28223 2/20 0.36
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
TAAR1 Q96RJ0 1/20 0.33
FOS P01100 1/20 0.33
TTR P02766 1/20 0.33
JUN P05412 1/20 0.33
NR3C1 P04150 1/20 0.33
HSD17B1 P14061 1/20 0.33
HSD17B2 P37059 1/20 0.33
S1PR1 P21453 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19446285 0.87 PTGS2 (0.39) PTGS2DHODHTRPM8
SCHEMBL12524837 0.84 PTGS2 (0.50) PTGS2HTR2AHTR2CHTR2BTAAR1
SCHEMBL19446284 0.81 PTGS2 (0.47) PTGS2HTR2AHTR2CHTR2BTAAR1
SCHEMBL15599161 0.78 S1PR1 (0.40) DHODHS1PR1
SCHEMBL10175179 0.77 TRPM8 (0.40) TRPM8S1PR1
SCHEMBL19446171 0.77 PTGS2 (0.43) PTGS2HTR2AHTR2CHTR2B
SCHEMBL188880 0.76 TRPM8 (0.39) TRPM8HTR2ATAAR1S1PR1
SCHEMBL10141662 0.76 TRPM8 (0.39) TRPM8S1PR1
SCHEMBL19446232 0.75 PTGS2 (0.38) PTGS2
SCHEMBL28484587 0.75 ABL1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2516417-B1 ISOINDOLINONE INHIBITORS OF PHOSPHATIDYLINOSITOL 3-KINASE VERTEX PHARMA (US) 2017-10-11 EP disclosed