Apovincamine

Apovincamine

SCHEMBL194507

CC[C@@]12C=C(C(=O)OC)n3c4c(c5ccccc53)CCN(CCC1)[C@H]42

nearest known ligand 0.85

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1A P54750 18/20 0.85
MEN1 O00255 2/20 0.85
LMNA P02545 2/20 0.85
KMT2A Q03164 2/20 0.85
HIF1A Q16665 2/20 0.85
CYP3A4 P08684 2/20 0.85
KDM4E B2RXH2 1/20 0.85
NR1I2 O75469 1/20 0.85
ALDH1A1 P00352 1/20 0.85
CHRM2 P08172 1/20 0.85
ADRA2A P08913 1/20 0.85
MAPT P10636 1/20 0.85
ADRA2B P18089 1/20 0.85
ADRA2C P18825 1/20 0.85
ADORA1 P30542 1/20 0.85
SLC6A4 P31645 1/20 0.85
DRD3 P35462 1/20 0.85
HTR2B P41595 1/20 0.85
BLM P54132 1/20 0.85
PDE1B Q01064 1/20 0.85

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Apovincamine SCHEMBL29421625 1.00 PDE1A (0.85) PDE1AMEN1LMNAKMT2AHIF1A
Apovincamine SCHEMBL10574604 1.00 PDE1A (0.85) PDE1AMEN1LMNAKMT2AHIF1A
Apovincamine SCHEMBL10571224 1.00 PDE1A (0.85) PDE1AMEN1LMNAKMT2AHIF1A
Apovincamine SCHEMBL11621460 0.96 PDE1A (0.79) PDE1AMEN1LMNAKMT2AHIF1A
Apovincamine SCHEMBL11619316 0.95 PDE1A (0.77) PDE1AMEN1LMNAKMT2AHIF1A
Apovincamine SCHEMBL11619228 0.92 PDE1A (0.72) PDE1AMEN1LMNAKMT2AHIF1A
Apovincamine SCHEMBL11619498 0.92 PDE1A (0.72) PDE1AMEN1LMNAKMT2AHIF1A
Apovincamine SCHEMBL11619109 0.92 PDE1A (0.72) PDE1AMEN1LMNAKMT2AHIF1A
Vinpocetine SCHEMBL7947532 0.92 PDE1A (1.00) PDE1AMEN1LMNAKMT2AHIF1A
Vinpocetine SCHEMBL21098929 0.92 PDE1A (1.00) PDE1AMEN1LMNAKMT2AHIF1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 410 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119548497-A Method for treating myopia by using vinpocetine 温州医科大学附属眼视光医院 2025-03-04 CN claimed
CN-118344985-A Genetically engineered bacterium for producing additional value products based on glucose, construction method and application 浙江大学杭州国际科创中心 2024-07-16 CN claimed
EP-4364736-A1 METHOD FOR TREATING MYOPIA WITH VINPOCETINE The Eye Hospital of Wenzhou Medical University (CN) 2024-05-08 EP claimed
WO-2023001176-A1 METHOD FOR TREATING MYOPIA WITH VINPOCETINE 温州医科大学附属眼视光医院 2023-01-26 WO claimed
CN-115634226-A Method for treating myopia by vinpocetine 温州医科大学附属眼视光医院 2023-01-24 CN claimed
US-20220233705-A1 COMBINED THERAPIES OF ACTIVATABLE IMMUNE CHECKPOINT INHIBITORS AND CONJUGATED ACTIVATABLE ANTIBODIES CYTOMX THERAPEUTICS INC (US) 2022-07-28 US claimed
CN-112649522-B Method for detecting related substances vinblastic acid and apovincamine acid in injection 海南葫芦娃药业集团股份有限公司 2022-02-22 CN claimed
EP-3930761-A1 COMBINED THERAPIES OF ACTIVATABLE IMMUNE CHECKPOINT INHIBITORS AND CONJUGATED ACTIVATABLE ANTIBODIES CytomX Therapeutics, Inc. (US) 2022-01-05 EP claimed
CN-113677372-A Combination therapy of activatable immune checkpoint inhibitors and conjugated activatable antibodies 西托姆克斯治疗公司 2021-11-19 CN claimed
CN-110950859-B Preparation method of vinpocetine 广州一品红制药有限公司 2021-04-30 CN claimed
EP-0573260-A1 New alkaloid derivatives, their use and pharmaceutical formulations containing them INDENA S.p.A. (IT) 1993-12-08 EP claimed
EP-0038619-B1 PROCESS FOR PREPARING VINCAMINE AND RELATED ALKALOIDS INVERNI DELLA BEFFA S.P.A. (IT) 1984-12-05 EP claimed
EP-0052238-B1 A NEW VINCAMINE DERIVATIVE, A METHOD FOR ITS PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING IT MEDEA RESEARCH S.r.l. (IT) 1984-05-09 EP claimed
EP-0045918-B1 A PROCESS FOR THE SYNTHESIS OF VINCAMINE AND RELATED INDOLE ALKALOIDS Mora, Paolo Corvi (IT) 1983-10-26 EP claimed
EP-0021923-B1 PROCESS FOR THE PREPARATION OF VINCAMINE DERIVATIVES SYNTHELABO (FR) 1983-09-07 EP claimed
EP-0052238-A1 A new vincamine derivative, a method for its preparation and pharmaceutical compositions containing it MEDEA RESEARCH S.r.l. (IT) 1982-05-26 EP claimed
US-4316029-A Synthesis of vincaminic acid derivatives SYNTHELABO (FR) 1982-02-16 US claimed
EP-0038619-A2 Process for preparing vincamine and related alkaloids INVERNI DELLA BEFFA S.P.A. (IT) 1981-10-28 EP claimed
EP-0021923-A1 Process for the preparation of vincamine derivatives SYNTHELABO (FR) 1981-01-07 EP claimed
US-4122179-A VASODILATORS Mora, Enrico Corvi (IT) 1978-10-24 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220233705-A1 COMBINED THERAPIES OF ACTIVATABLE IMMUNE CHECKPOINT INHIBITORS AND CONJUGATED ACTIVATABLE ANTIBODIES CD274, PDCD1LG2, PDCD1 PDE1A 1988/4885MEN1 1919/4885LMNA 3403/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.