SCHEMBL19454258

SCHEMBL19454258

O=C1NCCc2cc(Cc3ccccc3)ccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP11 Q9NR21 10/20 1.00
PARP10 Q53GL7 9/20 0.61
GRM5 P41594 7/20 0.57
PDPK1 O15530 1/20 0.56
PARP1 P09874 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10168733 0.80 PARP11 (0.66) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL25947316 0.80 PARP11 (0.66) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL8870301 0.78 PARP11 (0.63) PARP11
SCHEMBL4415080 0.77 MAOB (0.64) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL1951410 0.77 PARP11 (0.63) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL24852650 0.77 IL4I1 (0.63) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL8155722 0.76 PARP11 (1.00) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL19386434 0.76 PARP11 (0.61) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL20627544 0.76 PARP11 (0.61) PARP11PARP10GRM5PDPK1PARP1
SCHEMBL18010818 0.76 TDP2 (0.63) PARP11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017174757-A1 TETRAHYDROISOQUINOLINE ESTROGEN RECEPTOR MODULATORS AND USES THEREOF F. HOFFMANN-LA ROCHE AG (CH) 2017-10-12 WO disclosed