SCHEMBL19475461

SCHEMBL19475461

Cc1ccc2c(C(=O)O)cc(-c3ccc(N)cc3)nc2c1

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.70
ALDH1A1 P00352 4/20 0.70
PDE10A Q9Y233 3/20 0.70
HSD17B10 Q99714 3/20 0.63
DHODH Q02127 7/20 0.59
EPRS1 P07814 1/20 0.59
LMNA P02545 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
POLB P06746 1/20 0.53
TP53 P04637 2/20 0.52
HIF1A Q16665 2/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
KMT2A Q03164 1/20 0.50
PTGES O14684 1/20 0.50
ALOX5 P09917 1/20 0.50
CYP2C9 P11712 1/20 0.50
HPGD P15428 1/20 0.50
CASP7 P55210 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8619265 0.87 KDM4E (0.81) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL19475436 0.84 DHODH (0.64) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL19475477 0.84 HIF1A (0.68) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL16921273 0.83 DHODH (0.80) KDM4EALDH1A1PDE10ADHODHEPRS1
SCHEMBL8240327 0.82 POLB (0.66) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL4017739 0.80 DHODH (0.80) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL29788466 0.80 DHODH (0.80) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL8321335 0.78 ALDH1A1 (0.79) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL1898810 0.77 KDM4E (1.00) KDM4EALDH1A1PDE10AHSD17B10DHODH
SCHEMBL3457907 0.77 ALDH1A1 (0.77) KDM4EALDH1A1PDE10AHSD17B10DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017184547-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF NEW YORK UNIVERSITY (US) 2017-10-26 WO disclosed