SCHEMBL19475477

SCHEMBL19475477

Nc1ccc(-c2cc(C(=O)O)c3ccc(Cl)cc3n2)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 2/20 0.68
HSD17B10 Q99714 2/20 0.68
PTGES O14684 1/20 0.68
ALDH1A1 P00352 1/20 0.68
ALOX5 P09917 1/20 0.68
CYP2C9 P11712 1/20 0.68
HPGD P15428 1/20 0.68
CASP7 P55210 1/20 0.68
DHODH Q02127 8/20 0.62
EPRS1 P07814 1/20 0.59
KDM4E B2RXH2 2/20 0.55
LMNA P02545 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
PDE10A Q9Y233 1/20 0.55
POLB P06746 1/20 0.53
TP53 P04637 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2C19 P33261 1/20 0.52
KMT2A Q03164 1/20 0.52
EIF4A1 P60842 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19475331 0.90 ALDH1A1 (0.84) HIF1AHSD17B10PTGESALDH1A1ALOX5
SCHEMBL1901263 0.87 KDM4E (0.72) HIF1AHSD17B10PTGESALDH1A1ALOX5
SCHEMBL31590457 0.86 PTGES (0.68) HIF1AHSD17B10PTGESALDH1A1ALOX5
SCHEMBL19475297 0.86 PTGES (0.60) HIF1AHSD17B10PTGESALDH1A1ALOX5
SCHEMBL19475436 0.84 DHODH (0.64) HIF1AHSD17B10ALDH1A1DHODHEPRS1
SCHEMBL19475461 0.84 KDM4E (0.70) HIF1AHSD17B10PTGESALDH1A1ALOX5
SCHEMBL16921273 0.83 DHODH (0.80) ALDH1A1HPGDDHODHEPRS1KDM4E
SCHEMBL31590856 0.82 PTGES (0.61) HIF1AHSD17B10PTGESALDH1A1ALOX5
SCHEMBL14286200 0.81 HSD17B10 (1.00) HIF1AHSD17B10PTGESALDH1A1ALOX5
SCHEMBL5529524 0.81 HSD17B10 (0.94) HIF1AHSD17B10PTGESALDH1A1ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017184547-A1 QUINOLINE COMPOUNDS AS MODULATORS OF RAGE ACTIVITY AND USES THEREOF NEW YORK UNIVERSITY (US) 2017-10-26 WO disclosed