Forodesine

Forodesine

SCHEMBL1949526

Cl.OC[C@H]1N[C@@H](c2c[nH]c3c(O)ncnc23)[C@H](O)[C@@H]1O

nearest known ligand 0.73

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PNP

The experimentally established mechanism targets of Forodesine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
PNP known ✓ P00491 9/20 0.73
MTAP Q13126 10/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Forodesine SCHEMBL8244721 0.99 PNP (0.75) PNPMTAP
Forodesine SCHEMBL15740230 0.99 PNP (0.75) PNPMTAP
Forodesine SCHEMBL506383 0.99 PNP (0.75) PNPMTAP
Forodesine SCHEMBL8407141 0.99 PNP (0.75) PNPMTAP
Hydrochloric Acid SCHEMBL4837679 0.89 PNP (0.63) PNPMTAP
Galidesivir SCHEMBL30477706 0.86 PNP (0.97) PNPMTAP
Galidesivir SCHEMBL29577672 0.86 PNP (0.97) PNPMTAP
Galidesivir SCHEMBL15525360 0.86 PNP (0.97) PNPMTAP
Galidesivir SCHEMBL4838048 0.86 PNP (0.97) PNPMTAP
Galidesivir SCHEMBL23102311 0.85 PNP (1.00) PNPMTAP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8853224-B2 Acyclic amine inhibitors of nucleoside phosphorylases and hydrolases INDUSTRIAL RESEARCH LIMITED (NZ) 2014-10-07 US disclosed
EP-2395005-A1 Acyclic amine inhibitors of nucleoside phosphorylases and hydrolases Industrial Research Limited (NZ) 2011-12-14 EP disclosed
US-20110130412-A1 Acyclic amine inhibitors of nucleoside phosphorylases and hydrolases BIOCRYST PHARMACEUTICALS, INC. 2011-06-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110130412-A1 Acyclic amine inhibitors of nucleoside phosphorylases and hydrolases PNP, TYMP, NTPCR PNP 1/4885MTAP 12/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.