SCHEMBL19505947

SCHEMBL19505947

CCc1cccc(CC)c1NC(=O)NS(=O)(=O)c1cc(C(C)(C)O)cs1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 7/20 0.47
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
IDH1 O75874 1/20 0.41
CACNA1C Q13936 2/20 0.38
SCN5A Q14524 2/20 0.38
ANPEP P15144 1/20 0.38
CA2 P00918 1/20 0.38
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20929925 0.92 NLRP3 (0.46) NLRP3MEN1ALDH1A1KMT2ACA2
SCHEMBL19505716 0.88 NLRP3 (0.47) NLRP3IDH1CA2
SCHEMBL19505713 0.88 NLRP3 (0.39) NLRP3CA2
SCHEMBL19505715 0.85 NLRP3 (0.37) NLRP3CA2
SCHEMBL6555753 0.84 NLRP3 (0.66) NLRP3
SCHEMBL19505946 0.83 NLRP3 (0.52) NLRP3CA2
SCHEMBL29551031 0.83 NLRP3 (0.52) NLRP3CA2
SCHEMBL20930017 0.82 NLRP3 (0.46) NLRP3IDH1CA2
SCHEMBL7622551 0.80 NLRP3 (0.60) NLRP3
SCHEMBL19506004 0.78 NLRP3 (0.48) NLRP3KMT2AIDH1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11760735-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-09-19 US disclosed
US-11760735-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-09-19 US disclosed
US-11760735-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2023-09-19 US disclosed
US-20230099258-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY IFM THERAPEUTICS, INC. 2023-03-30 US disclosed
US-11339136-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2022-05-24 US disclosed
US-11339136-B2 Compounds and compositions for treating conditions associated with NLRP activity NOVARTIS AG (CH) 2022-05-24 US disclosed
EP-3445757-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RES INC (US) 2020-11-25 EP disclosed
EP-3445757-B1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS INFLAMMASOME RES INC (US) 2020-11-25 EP disclosed
US-20190119224-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2019-04-25 US disclosed
US-20190119224-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NOVARTIS AG (CH) 2019-04-25 US disclosed
WO-2017184624-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY IFM THERAPEUTICS, INC (US) 2017-10-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230099258-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 NLRP3 2/4885MEN1 3469/4885ALDH1A1 2031/4885
US-11760735-B2 Compounds and compositions for treating conditions associated with NLRP activity NLRP1, NLRP3, NOD1 NLRP3 2/4885MEN1 3469/4885ALDH1A1 2031/4885
US-20190119224-A1 COMPOUNDS AND COMPOSITIONS FOR TREATING CONDITIONS ASSOCIATED WITH NLRP ACTIVITY NLRP1, NLRP3, NOD1 NLRP3 2/4885MEN1 3469/4885ALDH1A1 2031/4885
US-11339136-B2 Compounds and compositions for treating conditions associated with NLRP activity NLRP1, NLRP3, NOD1 NLRP3 2/4885MEN1 3469/4885ALDH1A1 2031/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.