SCHEMBL19523402

SCHEMBL19523402

C=C(CNCCn1nc(-c2ccc(Oc3ccccc3)cc2)c2c(N)ncnc21)C(C)=O

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BTK Q06187 19/20 0.69
LCK P06239 8/20 0.69
EGFR P00533 6/20 0.69
ITK Q08881 6/20 0.69
JAK3 P52333 4/20 0.69
NUDT14 O95848 1/20 0.59
NUDT5 Q9UKK9 1/20 0.59
FYN P06241 3/20 0.51
LYN P07948 3/20 0.51
HCK P08631 3/20 0.51
FGR P09769 3/20 0.51
SRC P12931 3/20 0.51
FLT3 P36888 3/20 0.51
MAP2K1 Q02750 3/20 0.51
PTK6 Q13882 3/20 0.51
BRAF P15056 3/20 0.51
YES1 P07947 2/20 0.51
BLK P51451 2/20 0.51
BMX P51813 2/20 0.51
MAP2K5 Q13163 2/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14617791 0.86 BTK (0.78) BTKLCKEGFRITKJAK3
SCHEMBL25069009 0.84 NUDT14 (0.69) BTKLCKEGFRITKJAK3
SCHEMBL15517319 0.84 BTK (0.81) BTKLCKEGFRITKJAK3
SCHEMBL17090646 0.83 BTK (0.80) BTKLCKEGFRITKJAK3
SCHEMBL22909341 0.82 NUDT14 (0.72) BTKLCKEGFRITKJAK3
SCHEMBL14643776 0.82 BTK (0.76) BTKLCKEGFRITKJAK3
SCHEMBL14617765 0.82 BTK (0.76) BTKLCKEGFRITKJAK3
SCHEMBL16701418 0.82 BTK (0.67) BTKLCKEGFRITKJAK3
SCHEMBL408564 0.81 BTK (1.00) BTKLCKEGFRITKJAK3
SCHEMBL14617775 0.81 BTK (0.80) BTKLCKEGFRITKJAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9801881-B2 Use of inhibitors of bruton's tyrosine kinase (BTK) PHARMACYCLICS LLC (US) 2017-10-31 US disclosed