SCHEMBL195519

SCHEMBL195519

O=C(O)c1cc(Br)c(Br)c(Br)c1C(=O)O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.42
AKR1C4 P17516 2/20 0.42
AKR1C2 P52895 2/20 0.42
AKR1C1 Q04828 2/20 0.42
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
TSHR P16473 2/20 0.39
PTPN1 P18031 3/20 0.38
EIF2AK2 P19525 1/20 0.38
CSNK2A2 P19784 1/20 0.38
CSNK2B P67870 1/20 0.38
CSNK2A1 P68400 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA3 P07451 1/20 0.38
CA4 P22748 1/20 0.38
CA6 P23280 1/20 0.38
CA5A P35218 1/20 0.38
CA7 P43166 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10434460 0.84 EIF2AK2 (0.38) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL22802151 0.83 TSHR (0.43) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL8941154 0.82 AKR1C4 (0.42) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL10868192 0.82 AKR1C4 (0.42) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL11678633 0.81 EIF2AK2 (0.41) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL49516 0.81 EIF2AK2 (0.45) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL17512444 0.81 LCK (0.33) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL28264157 0.79 TSHR (0.40) AKR1C3AKR1C4AKR1C2AKR1C1LCK
SCHEMBL30555489 0.77 AKR1C3 (0.57) AKR1C3AKR1C4AKR1C2AKR1C1PTPN1
SCHEMBL605556 0.77 AKR1C3 (0.57) AKR1C3AKR1C4AKR1C2AKR1C1PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7611572-B2 Pixel-forming colorant compositions and their use DAINICHISEIKA COLOR & CHEMICALS MFG. CO., LTD. (JP) 2009-11-03 US claimed
EP-1717277-A2 Pixel-forming colorant compositions and their use Dainichiseika Color & Chemicals Mfg. Co., Ltd. (JP) 2006-11-02 EP claimed
US-20060213394-A1 PIXEL-FORMING COLORANT COMPOSITIONS AND THEIR USE DAINICHISEIKA COLOR & CHEMICALS MFG. CO., LTD. (JP) 2006-09-28 US claimed
US-6190581-B1 MIXING SODIUM ANTIMONATE HYDRATE WITH A POLYMER AND ADDING TO VENTED OR VACUUM APPARATUS OR HIGH SHEAR BLENDER AT GIVEN HIGH TEMPERATURE RANGE TO PRODUCE A FLAMEPROOFING CONCENTRATE FOR ADDITION TO A POLYMER SUCH AS POLYETHYLENE TEREPHTHALATE LAUREL INDUSTRIES, INC. 2001-02-20 US claimed
EP-1717277-B1 Pixel-forming colorant compositions and their use DAINICHISEIKA COLOR CHEM (JP) 2012-01-04 EP disclosed
US-7611572-B2 Pixel-forming colorant compositions and their use DAINICHISEIKA COLOR & CHEMICALS MFG. CO., LTD. (JP) 2009-11-03 US disclosed
US-20060292450-A1 Non-aqueous electrolyte secondary battery MATSUSHITA ELECTRIC INDUSTRIAL CO., LTD. 2006-12-28 US disclosed
EP-1717277-A2 Pixel-forming colorant compositions and their use Dainichiseika Color & Chemicals Mfg. Co., Ltd. (JP) 2006-11-02 EP disclosed
US-20060213394-A1 PIXEL-FORMING COLORANT COMPOSITIONS AND THEIR USE DAINICHISEIKA COLOR & CHEMICALS MFG. CO., LTD. (JP) 2006-09-28 US disclosed
US-6797760-B1 Non-dripping, flame retardant, fluoroelastomer insulative compositions for telecommunication cables ALPHAGARY CORPORATION 2004-09-28 US disclosed
WO-2001046311-A1 ESTERIFICATION METHOD TEKNOR APEX COMPANY (US) 2001-06-28 WO disclosed
US-6232427-B1 MIXTURE OF POLYMER AND PLASTICIZER TEKNOR APEX COMPANY 2001-05-15 US disclosed
US-6190581-B1 MIXING SODIUM ANTIMONATE HYDRATE WITH A POLYMER AND ADDING TO VENTED OR VACUUM APPARATUS OR HIGH SHEAR BLENDER AT GIVEN HIGH TEMPERATURE RANGE TO PRODUCE A FLAMEPROOFING CONCENTRATE FOR ADDITION TO A POLYMER SUCH AS POLYETHYLENE TEREPHTHALATE LAUREL INDUSTRIES, INC. 2001-02-20 US disclosed
WO-1999029778-A1 ESTERIFICATION METHOD TEKNOR APEX COMPANY (US) 1999-06-17 WO disclosed
US-4002642-A Process for the preparation of polyhalo copper phthalocyanines HOECHST AKTIENGESELLSCHAFT (DT) 1977-01-11 US disclosed