SCHEMBL19557281

SCHEMBL19557281

CC[Si](CC)(CC)c1cc2ccccc2n1COCC[Si](C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.42
DGAT1 O75907 2/20 0.34
MTNR1A P48039 3/20 0.32
MTNR1B P49286 3/20 0.32
TP53 P04637 2/20 0.32
TSHR P16473 1/20 0.32
EGFR P00533 1/20 0.32
IGF1R P08069 1/20 0.32
SRC P12931 1/20 0.32
FLT4 P35916 1/20 0.32
KDR P35968 1/20 0.32
FLT3 P36888 1/20 0.32
EPHB4 P54760 1/20 0.32
TEK Q02763 1/20 0.32
F11 P03951 1/20 0.31
MAPT P10636 1/20 0.31
KDM4E B2RXH2 3/20 0.31
HPGD P15428 2/20 0.31
ALDH1A1 P00352 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29287219 0.81 NPC1 (0.46) NPC1TP53TSHRMAPTKDM4E
SCHEMBL29509222 0.80 KDM4E (0.43) NPC1MTNR1AMTNR1BTP53TSHR
SCHEMBL17504855 0.80 KDM4E (0.43) NPC1MTNR1AMTNR1BTP53TSHR
SCHEMBL19492427 0.80 NPC1 (0.45) NPC1DGAT1MTNR1AMTNR1BTP53
SCHEMBL17504852 0.78 NPC1 (0.42) NPC1MTNR1AMTNR1BTP53TSHR
SCHEMBL29509131 0.78 NPC1 (0.42) NPC1MTNR1AMTNR1BTP53TSHR
SCHEMBL19557279 0.77 HTT (0.42) NPC1TP53TSHRMAPTKDM4E
SCHEMBL19463815 0.76 NPC1 (0.45) NPC1DGAT1MTNR1AMTNR1BTP53
SCHEMBL14498914 0.76 NPC1 (0.42) NPC1DGAT1MTNR1AMTNR1BTP53
SCHEMBL30455806 0.76 NPC1 (0.45) NPC1DGAT1MTNR1AMTNR1BTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11753421-B2 Silylated derivatives of aromatic heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2023-09-12 US disclosed
US-11753421-B2 Silylated derivatives of aromatic heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2023-09-12 US disclosed
CN-111253424-B Silylation of aromatic heterocycles over earth-rich transition metal-free catalysts 加州理工学院 2023-06-20 CN disclosed
EP-3705482-B1 SILYLATION OF AROMATIC HETEROCYCLES BY EARTH ABUNDANT TRANSITION-METAL-FREE CATALYSTS CALIFORNIA INST OF TECHN (US) 2023-02-22 EP disclosed
US-20220185828-A1 Silylated Derivatives Of Aromatic Heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY 2022-06-16 US disclosed
US-11312733-B2 Silylated derivatives of aromatic heterocycles CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2022-04-26 US disclosed
CN-111253424-A Silylation of aromatic heterocycles by earth-rich transition metal-free catalysts 加州理工学院 2020-06-09 CN disclosed
CN-107108662-B9 Silylation of aromatic heterocycles by earth-rich transition metal-free catalysts 加州理工学院 2020-05-15 CN disclosed
CN-107108662-B Silylation of aromatic heterocycles by earth-rich transition metal-free catalysts 加州理工学院 2020-02-07 CN disclosed
US-20180057514-A1 SILYLATION OF AROMATIC HETEROCYCLES BY EARTH ABUNDANT TRANSITION-METAL-FREE CATALYSTS CALIFORNIA INSTITUTE OF TECHNOLOGY 2018-03-01 US disclosed
US-9809607-B2 Silylation of aromatic heterocycles by earth abundant transition-metal-free catalysts CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2017-11-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11312733-B2 Silylated derivatives of aromatic heterocycles KCNH1, KCNH3, HNRNPH3 NPC1 1172/4885DGAT1 4477/4885MTNR1A 4703/4885
US-20180057514-A1 SILYLATION OF AROMATIC HETEROCYCLES BY EARTH ABUNDANT TRANSITION-METAL-FREE CATALYSTS TEC, AURKA, TYR NPC1 1990/4885DGAT1 3865/4885MTNR1A 4705/4885
US-11753421-B2 Silylated derivatives of aromatic heterocycles KCNH1, KCNH3, HNRNPH3 NPC1 1172/4885DGAT1 4477/4885MTNR1A 4703/4885
US-20220185828-A1 Silylated Derivatives Of Aromatic Heterocycles KCNH1, KCNH3, HNRNPH3 NPC1 1172/4885DGAT1 4477/4885MTNR1A 4703/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.