SCHEMBL19583237

SCHEMBL19583237

Cn1c(=O)c2[nH]c(Cl)nc2n(CCC2CC2)c1=O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 2/20 0.44
PDE1A P54750 2/20 0.44
PDE1B Q01064 2/20 0.44
PDE1C Q14123 2/20 0.44
PDE5A O76074 1/20 0.44
PDE4A P27815 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
ADORA1 P30542 5/20 0.43
ADORA2A P29274 4/20 0.43
ADORA2B P29275 3/20 0.43
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
ADORA3 P0DMS8 1/20 0.42
NFKB1 P19838 1/20 0.42
MAPK1 P28482 1/20 0.42
PMP22 Q01453 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13533471 0.86 PDE5A (0.49) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL3175238 0.83 PDE4A (0.43) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL3123904 0.82 ADORA2A (0.46) PDE4APDE4BPDE4CPDE4DADORA1
SCHEMBL3175170 0.82 PDE4A (0.55) PDE4APDE4BPDE4CPDE4DADORA2A
SCHEMBL1808708 0.81 PDE1A (0.48) PDE2APDE1APDE1BPDE1CPDE5A
SCHEMBL3181178 0.80 ADORA2A (0.54) PDE2APDE1APDE1BPDE1CPDE5A
SCHEMBL3119502 0.80 ADORA1 (0.47) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL3175131 0.80 PDE4A (0.57) PDE2APDE1APDE1BPDE1CPDE4A
SCHEMBL3185628 0.78 ADORA1 (0.48) PDE4APDE4BPDE4CPDE4DADORA1
SCHEMBL19583228 0.78 PDE1A (0.56) PDE2APDE1APDE1BPDE1CPDE5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3251675-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE Shanton Pharma Co., Ltd. (CN) 2017-12-06 EP claimed
US-20170326148-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE Shanton Pharma Pte. Ltd. (SG) 2017-11-16 US claimed
EP-3251675-B1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE SHANTON PHARMA PTE LTD (SG) 2021-04-21 EP disclosed
US-10322132-B2 Prevention or treatment of uratic or gouty diseases SHANTON PHARMA CO., LTD (CN) 2019-06-18 US disclosed
EP-3251675-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE Shanton Pharma Co., Ltd. (CN) 2017-12-06 EP disclosed
US-20170326148-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE Shanton Pharma Pte. Ltd. (SG) 2017-11-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170326148-A1 PREVENTION OR TREATMENT OF URIC ACID OR GOUT DISEASE NLRP3, REN, SLC5A1 PDE2A 2077/4885PDE1A 4787/4885PDE1B 4808/4885
US-10322132-B2 Prevention or treatment of uratic or gouty diseases REN, NLRP3, SLC5A1 PDE2A 2454/4885PDE1A 4751/4885PDE1B 4795/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.