SCHEMBL19611005

SCHEMBL19611005

C[C@H]1CCCC[C@H]1NC(=O)Oc1cc2ccc(Br)cc2[nH]1

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 1/20 0.44
TAS1R3 Q7RTX0 11/20 0.41
TAS1R1 Q7RTX1 10/20 0.41
TAS1R2 Q8TE23 9/20 0.41
CHRNA7 P36544 1/20 0.40
HPGD P15428 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ALDH1A1 P00352 3/20 0.38
LMNA P02545 2/20 0.38
USP2 O75604 1/20 0.38
POLB P06746 1/20 0.38
RECQL P46063 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19610999 0.88 TAS1R3 (0.44) TAS1R3TAS1R1TAS1R2L3MBTL1ALDH1A1
SCHEMBL19611046 0.84 TAS1R3 (0.39) TAS1R3TAS1R1TAS1R2ALDH1A1LMNA
SCHEMBL19610988 0.81 TAS1R3 (0.42) TAS1R3TAS1R1TAS1R2CHRNA7HPGD
SCHEMBL15506751 0.81 DRD4 (0.65) DRD4TAS1R3TAS1R1TAS1R2ALDH1A1
SCHEMBL19611049 0.79 ALDH1A1 (0.44) TAS1R3TAS1R1TAS1R2L3MBTL1ALDH1A1
SCHEMBL19611022 0.77 TAS1R3 (0.45) TAS1R3TAS1R1TAS1R2CHRNA7ALDH1A1
SCHEMBL19611026 0.76 TAS1R3 (0.48) TAS1R3TAS1R1TAS1R2HPGDL3MBTL1
SCHEMBL19611031 0.74 TAS1R3 (0.52) TAS1R3TAS1R1TAS1R2HPGDL3MBTL1
SCHEMBL19610986 0.74 TAS1R3 (0.52) TAS1R3TAS1R1TAS1R2HPGDL3MBTL1
SCHEMBL19611051 0.74 TAS1R3 (0.52) TAS1R3TAS1R1TAS1R2HPGDL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2892880-B1 INDOLE CARBOXAMIDE DERIVATIVES AND USES THEREOF NOVARTIS AG (CH) 2017-11-22 EP claimed