SCHEMBL19611883

SCHEMBL19611883

Nc1cccc2c1C(=O)N(C1CCCC(=O)NC1=O)C2=O

nearest known ligand 0.85

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 17/20 0.85
DDB1 Q16531 16/20 0.85
IKZF3 Q9UKT9 3/20 0.85
TNF P01375 2/20 0.85
IL1B P01584 2/20 0.85
IKZF1 Q13422 2/20 0.85
TBXA2R P21731 1/20 0.85
ALDH1A1 P00352 1/20 0.62
CHRM2 P08172 1/20 0.62
OPRM1 P35372 1/20 0.62
CYP1A2 P05177 1/20 0.62
TSHR P16473 1/20 0.62
TDP1 Q9NUW8 1/20 0.62
BRD4 O60885 1/20 0.53
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HTR3E A5X5Y0 1/20 0.52
HTR3B O95264 1/20 0.52
HTR2B P41595 1/20 0.52
HTR3A P46098 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18263919 1.00 CRBN (0.85) CRBNDDB1IKZF3TNFIL1B
SCHEMBL18263946 1.00 CRBN (0.85) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL15930059 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL19250920 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL29382107 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL15930065 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL369172 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL931134 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL563317 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B
Pomalidomide SCHEMBL15930061 0.92 CRBN (1.00) CRBNDDB1IKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11773080-B2 Deuterium-enriched isoindolinonyl-azepanediones and related compounds and methods of treating medical disorders using same SALARIUS PHARMACEUTICALS, INC. (US) 2023-10-03 US disclosed
US-20210340125-A1 DEUTERIUM-ENRICHED ISOINDOLINONYL-AZEPANEDIONES AND RELATED COMPOUNDS AND METHODS OF TREATING MEDICAL DISORDERS USING SAME SALARIUS PHARMACEUTICALS, INC. 2021-11-04 US disclosed
US-10562917-B2 Chimeric compounds targeting proteins, compositions, methods, and uses thereof BIOTHERYX, INC. (US) 2020-02-18 US disclosed
US-20190276474-A1 CHIMERIC COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF BIOTHERYX, INC. 2019-09-12 US disclosed
US-10144745-B2 Chimeric compounds targeting proteins, compositions, methods, and uses thereof BIOTHERYX, INC. (US) 2018-12-04 US disclosed
US-9938302-B2 Chimeric compounds targeting proteins, compositions, methods, and uses thereof BIOTHERYX, INC. (US) 2018-04-10 US disclosed
US-20170334932-A1 CHIMERIC COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF BIOTHERYX, INC. 2017-11-23 US disclosed
US-20170333443-A1 CHIMERIC COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF BIOTHERYX, INC. 2017-11-23 US disclosed
WO-2017201069-A1 OXOINDOLINE DERIVATIVES AS PROTEIN FUNCTION MODULATORS BIOTHERYX, INC. (US) 2017-11-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10144745-B2 Chimeric compounds targeting proteins, compositions, methods, and uses thereof IKZF3, IKZF1, CKS1B CRBN 176/4885DDB1 2485/4885IKZF3 1/4885
US-11773080-B2 Deuterium-enriched isoindolinonyl-azepanediones and related compounds and methods of treating medical disorders using same HPGDS, HPGD, AQP3 CRBN 1079/4885DDB1 690/4885IKZF3 318/4885
US-10562917-B2 Chimeric compounds targeting proteins, compositions, methods, and uses thereof IKZF3, IKZF1, CKS1B CRBN 176/4885DDB1 2485/4885IKZF3 1/4885
US-20210340125-A1 DEUTERIUM-ENRICHED ISOINDOLINONYL-AZEPANEDIONES AND RELATED COMPOUNDS AND METHODS OF TREATING MEDICAL DISORDERS USING SAME HPGDS, HPGD, AQP3 CRBN 1079/4885DDB1 690/4885IKZF3 318/4885
US-20170333443-A1 CHIMERIC COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF IKZF3, IKZF1, CKS1B CRBN 176/4885DDB1 2485/4885IKZF3 1/4885
US-20170334932-A1 CHIMERIC COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF IKZF3, IKZF1, CKS1B CRBN 176/4885DDB1 2485/4885IKZF3 1/4885
US-20190276474-A1 CHIMERIC COMPOUNDS TARGETING PROTEINS, COMPOSITIONS, METHODS, AND USES THEREOF IKZF3, IKZF1, CKS1B CRBN 176/4885DDB1 2485/4885IKZF3 1/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.