SCHEMBL1961206

SCHEMBL1961206

Clc1ccc(Br)c(Br)c1Cl

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.38
MAPK1 P28482 1/20 0.38
CYP2A6 P11509 2/20 0.33
AHR P35869 2/20 0.32
CXCR1 P25024 1/20 0.32
CXCR2 P25025 1/20 0.32
TDP1 Q9NUW8 1/20 0.31
TSHR P16473 1/20 0.31
CYP1A2 P05177 2/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
CYP2D6 P10635 1/20 0.30
NFKB1 P19838 1/20 0.30
PNMT P11086 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10875349 0.81 CYP3A4 (0.41) CYP3A4MAPK1CYP2A6AHRTDP1
SCHEMBL11177494 0.79 CYP1A2 (0.32) CYP2A6AHRTSHRCYP1A2HTR2A
SCHEMBL1446088 0.79 CYP3A4 (0.46) CYP3A4MAPK1CYP2A6AHRCXCR1
SCHEMBL23273230 0.77 HTR2A (0.34) CYP3A4MAPK1CYP2A6TDP1CYP1A2
SCHEMBL1561688 0.72 CYP3A4 (0.35) CYP3A4MAPK1CYP2A6AHRCXCR1
SCHEMBL11595170 0.72 CYP3A4 (0.59) CYP3A4MAPK1CXCR1CXCR2TDP1
SCHEMBL7615955 0.72 CYP3A4 (0.35) CYP3A4MAPK1CYP2A6AHRCXCR1
SCHEMBL19830027 0.72 CYP3A4 (0.36) CYP3A4MAPK1CYP2A6AHRHTR2A
SCHEMBL10990892 0.72 TSHR (0.39) CYP3A4MAPK1AHRTDP1TSHR
SCHEMBL4448667 0.72 ALDH1A1 (0.36) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 169 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20010039349-A1 Selective, Catalytic, thermal functionalization of secondary or aromatic C-H cyclic hydrocarbon bonds SHELL OIL COMPANY 2001-11-08 US claimed
US-4347390-A Process for producing 1-bromo-3,5-dichlorobenzene ISHIHARA SANGYO KAISHA LTD. 1982-08-31 US claimed
US-9115151-B2 Substituted 2,10-dihydro-9-oxa-1,2,4A-triazaphenanthren-3-ones and uses thereof ABBVIE INC. (US) 2015-08-25 US disclosed
US-9115151-B2 Substituted 2,10-dihydro-9-oxa-1,2,4A-triazaphenanthren-3-ones and uses thereof ABBVIE INC. (US) 2015-08-25 US disclosed
CN-102712704-B Three and four atom bridged dicarbonate compounds as internal donors in catalysts for polypropylene manufacture DOW GLOBAL TECHNOLOGIES INC 2015-01-07 CN disclosed
CN-102762603-B Two atom bridged dicarbonate compounds as internal donors in catalysts for polypropylene manufacture DOW GLOBAL TECHNOLOGIES LLC (US) 2014-11-26 CN disclosed
EP-2507269-B1 THREE AND FOUR ATOM BRIDGED DICARBONATE COMPOUNDS AS INTERNAL DONORS IN CATALYSTS FOR POLYPROPYLENE MANUFACTURE GRACE W R & CO (US) 2014-10-29 EP disclosed
EP-2507268-B1 TWO ATOM BRIDGED DICARBONATE COMPOUNDS AS INTERNAL DONORS IN CATALYSTS FOR POLYPROPYLENE MANUFACTURE GRACE W R & CO (US) 2014-10-15 EP disclosed
US-20140206663-A1 TRIAZINONE COMPOUNDS WUXI APPTECH (SHANGHAI) CO., LTD. (CN) 2014-07-24 US disclosed
US-20140206663-A1 TRIAZINONE COMPOUNDS WUXI APPTECH (SHANGHAI) CO., LTD. (CN) 2014-07-24 US disclosed
WO-2014089904-A1 TRIAZINONE COMPOUNDS ABBVIE INC. (US) 2014-06-19 WO disclosed
US-4414132-A Olefin polymerization catalyst compositions and a process for the polymerization of olefins employing such compositions SHELL OIL COMPANY (US) 1983-11-08 US disclosed
EP-0019330-B1 OLEFIN POLYMERIZATION CATALYST COMPOSITIONS AND A PROCESS FOR THE POLYMERIZATION OF OLEFINS EMPLOYING SUCH COMPOSITIONS SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1983-08-31 EP disclosed
US-4400302-A TITANIUM HALIDE, ALKYL MAGNESIUM SHELL OIL COMPANY (US) 1983-08-23 US disclosed
EP-0046859-B1 PROCESS FOR THE PREPARATION OF 1-BROMO-3,5-DICHLOROBENZENE BASF Aktiengesellschaft (DE) 1983-07-06 EP disclosed
US-4368340-A VAPOR PHASE CHLORINATION OF 1,3,5-TRIHALOBENZENE HAVING BROMINE ATOMS ISHIHARA SANGYO KAISHA LTD. (JP) 1983-01-11 US disclosed
EP-0063066-A1 Process for the isomerization of bromohalogen benzenes RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1982-10-20 EP disclosed
US-4347390-A Process for producing 1-bromo-3,5-dichlorobenzene ISHIHARA SANGYO KAISHA LTD. 1982-08-31 US disclosed
EP-0046859-A1 Process for the preparation of 1-bromo-3,5-dichlorobenzene BASF Aktiengesellschaft (DE) 1982-03-10 EP disclosed
EP-0019330-A1 Olefin polymerization catalyst compositions and a process for the polymerization of olefins employing such compositions SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1980-11-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140206663-A1 TRIAZINONE COMPOUNDS THPO, IL5, CYP11B2 CYP3A4 21/4885MAPK1 1200/4885CYP2A6 60/4885
US-20010039349-A1 Selective, Catalytic, thermal functionalization of secondary or aromatic C-H cyclic hydrocarbon bonds AHR, PAH, HRH3 CYP3A4 125/4885MAPK1 2544/4885CYP2A6 284/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.