SCHEMBL19619488

SCHEMBL19619488

CC(C)c1ccc(C(C)(F)P)nc1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.39
CHRNA7 P36544 2/20 0.35
HSD11B1 P28845 1/20 0.34
PDE2A O00408 1/20 0.32
P2RX7 Q99572 1/20 0.32
NR1I2 O75469 1/20 0.31
CYP2C9 P11712 1/20 0.31
PTPN5 P54829 1/20 0.31
MLYCD O95822 2/20 0.31
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18570673 0.89 TRPV4 (0.39) TRPV4CHRNA7HSD11B1PTPN5MLYCD
SCHEMBL17775927 0.86 TRPV4 (0.36) TRPV4CHRNA7HSD11B1PDE2ANR1I2
SCHEMBL17775982 0.86 TRPV4 (0.36) TRPV4CHRNA7HSD11B1PDE2ANR1I2
SCHEMBL21076643 0.85 TRPV4 (0.37) TRPV4CHRNA7HSD11B1
SCHEMBL2609310 0.84 TRPV4 (0.52) TRPV4CHRNA7HSD11B1PDE2AP2RX7
SCHEMBL26326434 0.83 CHRNA7 (0.35) TRPV4CHRNA7
SCHEMBL20390072 0.83 CHRNA7 (0.35) TRPV4CHRNA7HSD11B1PDE2ANR1I2
SCHEMBL20390073 0.83 CHRNA7 (0.35) TRPV4CHRNA7HSD11B1PDE2ANR1I2
SCHEMBL1694606 0.82 CHRNA7 (0.38) TRPV4CHRNA7HSD11B1NR1I2CYP2C9
SCHEMBL20392645 0.81 CHRNA7 (0.35) TRPV4CHRNA7HSD11B1PDE2APTPN5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9822130-B2 Triazolo-pyrazinyl derivatives useful as soluble guanylate cyclase activators MERCK SHARP & DOHME CORP. (US) 2017-11-21 US disclosed