SCHEMBL19620492

SCHEMBL19620492

NC1=C(OSCc2ccccc2)C(=O)C(c2ccc(Cl)c(Cl)c2)O1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
KCNA5 P22460 1/20 0.36
ADK P55263 3/20 0.35
SLC6A2 P23975 7/20 0.34
SLC6A3 Q01959 7/20 0.34
F10 P00742 1/20 0.33
SLC6A4 P31645 4/20 0.32
PPARG P37231 2/20 0.32
NPSR1 Q6W5P4 1/20 0.32
NR2E3 Q9Y5X4 1/20 0.32
NCOR2 Q9Y618 1/20 0.32
EDNRA P25101 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C19 P33261 1/20 0.31
PPARA Q07869 1/20 0.30
BACE1 P56817 1/20 0.30
FFAR1 O14842 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19620572 0.90 KDM4E (0.34) KDM4EPOLBMAPTADK
SCHEMBL19620596 0.90 KDM4E (0.34) KDM4EPOLBMAPTADKSLC6A2
SCHEMBL19620522 0.87 KDM4E (0.42) KDM4EPOLBMAPTKCNA5ADK
SCHEMBL19620570 0.86 MAPT (0.39) KDM4EPOLBMAPTSLC6A3
SCHEMBL19620689 0.86 KDM4E (0.38) KDM4EPOLBMAPTADKCYP1A2
SCHEMBL19620603 0.85 POLB (0.50) KDM4EPOLBMAPTADKSLC6A3
SCHEMBL19620589 0.85 ADK (0.39) KDM4EPOLBMAPTADKSLC6A2
SCHEMBL19620593 0.84 KDM4E (0.36) KDM4EPOLBMAPTADKCYP1A2
SCHEMBL19620669 0.83 CYP1A2 (0.34) KDM4EPOLBMAPTNPSR1CYP1A2
SCHEMBL19620542 0.82 POLB (0.42) KDM4EPOLBMAPTADKSLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2897607-B1 INHIBITORS OF BETA-HYDROLASE FOR TREATMENT OF CANCER RHODE ISLAND HOSPITAL (US) 2017-11-22 EP disclosed