SCHEMBL19622253

SCHEMBL19622253

CCC(=O)Oc1ccc(Oc2ccc3c(c2)COB3)c(Oc2ccc(C#N)cn2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 4/20 0.43
HRH3 Q9Y5N1 1/20 0.36
SCN9A Q15858 4/20 0.35
FPR2 P25090 1/20 0.35
SCN7A Q01118 3/20 0.33
KCNH2 Q12809 3/20 0.33
P2RX3 P56373 2/20 0.32
PANK3 Q9H999 1/20 0.32
OPRM1 P35372 1/20 0.32
PPARD Q03181 2/20 0.32
PPARA Q07869 2/20 0.32
CHRM1 P11229 1/20 0.32
PDE4A P27815 1/20 0.32
ADRA1A P35348 1/20 0.32
PDE1A P54750 1/20 0.32
PDE4C Q08493 1/20 0.32
PDE4D Q08499 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE7A Q13946 1/20 0.32
PDE3A Q14432 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8004246 0.81 PDE4B (0.58) PDE4BHRH3SCN9AFPR2SCN7A
SCHEMBL19622217 0.80 FGFR1 (0.39)
SCHEMBL8010823 0.79 PDE4B (0.42) PDE4BHRH3SCN9AFPR2OPRM1
SCHEMBL19622216 0.77 ACHE (0.36)
SCHEMBL14748446 0.74 PTGDR2 (0.45) PDE4BPPARDPPARACHRM1PDE4A
SCHEMBL14748461 0.73 TBXA2R (0.36) PDE4BPPARDPPARACHRM1PDE4A
SCHEMBL8005546 0.72 AR (0.59) PDE4BKCNH2PPARDPPARACHRM1
SCHEMBL19622265 0.72 AR (0.36) PDE4BSCN9APPARDPPARACHRM1
SCHEMBL8005549 0.71 AR (0.44) PDE4BKCNH2CHRM1PDE4AADRA1A
SCHEMBL7862450 0.70 PDE4B (0.43) PDE4BPDE4APDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed