SCHEMBL19622296

SCHEMBL19622296

N#Cc1ccc(Oc2ccc3c(c2)CO3)cc1Cl

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AR P10275 2/20 0.48
PGR P06401 3/20 0.44
PDE4B Q07343 1/20 0.44
SLC22A12 Q96S37 13/20 0.42
TRPV4 Q9HBA0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19622248 0.83 PDE4B (0.44) ARPDE4BSLC22A12
SCHEMBL7997145 0.77 AR (0.45) ARPGRPDE4BSLC22A12TRPV4
SCHEMBL4181007 0.77 AR (0.50) ARPGRPDE4BSLC22A12TRPV4
SCHEMBL2526722 0.75 PDE4B (0.79) PDE4B
SCHEMBL8543199 0.75 AR (0.62) ARPGRSLC22A12TRPV4
SCHEMBL4184922 0.73 AR (0.65) ARPGRSLC22A12TRPV4
SCHEMBL13890483 0.73 AR (0.56) ARPGRPDE4BSLC22A12TRPV4
SCHEMBL1656135 0.72 PDE4B (0.51) ARPDE4B
SCHEMBL474005 0.72 AR (0.68) ARPGRSLC22A12TRPV4
SCHEMBL4171343 0.72 AR (0.59) ARPGRSLC22A12TRPV4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed