SCHEMBL19622248

SCHEMBL19622248

Cc1cc(Oc2ccc3c(c2)CO3)ccc1C#N

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 5/20 0.44
AR P10275 10/20 0.41
SLC22A12 Q96S37 1/20 0.39
ESRRA P11474 1/20 0.37
PDE4A P27815 2/20 0.36
PDE4C Q08493 2/20 0.36
PDE4D Q08499 2/20 0.36
CHRM1 P11229 1/20 0.36
ADRA1A P35348 1/20 0.36
PDE1A P54750 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE7A Q13946 1/20 0.36
PDE3A Q14432 1/20 0.36
MRGPRX4 Q96LA9 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19622296 0.83 AR (0.48) PDE4BARSLC22A12
SCHEMBL2531105 0.75 PDE4B (0.79) PDE4BPDE4APDE4CPDE4DCHRM1
SCHEMBL13890548 0.73 AR (0.53) PDE4BARPDE4APDE4CPDE4D
SCHEMBL17623897 0.73 AR (0.53) ARMRGPRX4
SCHEMBL1656135 0.72 PDE4B (0.51) PDE4BAR
SCHEMBL4377219 0.72 AR (0.53) ARSLC22A12
SCHEMBL509379 0.69 AR (0.50) ARMRGPRX4
SCHEMBL25865448 0.69 AR (0.48) ARMRGPRX4
SCHEMBL13890508 0.68 AR (0.66) PDE4BARSLC22A12PDE4APDE4C
SCHEMBL25680960 0.68 AR (0.44) ARSLC22A12ESRRAMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3246034-A1 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS Anacor Pharmaceuticals, Inc. (US) 2017-11-22 EP disclosed