SCHEMBL19623807

SCHEMBL19623807

O=Nc1ccc(NCCCN2CCOCC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.51
RAB9A P51151 3/20 0.51
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
RAD52 P43351 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
MAPT P10636 3/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
KDM4E B2RXH2 2/20 0.47
POLB P06746 2/20 0.47
GAA P10253 2/20 0.47
LMNA P02545 1/20 0.47
GLA P06280 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
HSD17B10 Q99714 1/20 0.46
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14262798 0.87 BACE1 (0.47) L3MBTL1MAPTCACNA1B
SCHEMBL14262613 0.84 KMT2A (0.43) RAB9AKMT2AMAPTLMNATSHR
SCHEMBL8243016 0.82 LMNA (0.58) NPC1RAB9AKMT2AMEN1RAD52
SCHEMBL1955959 0.81 NPC1 (0.51) NPC1RAB9AKMT2AMEN1RAD52
SCHEMBL3234489 0.81 NPC1 (0.51) NPC1RAB9AKMT2AMEN1RAD52
SCHEMBL19623580 0.81 RAD52 (0.53) NPC1RAB9AKMT2AMEN1RAD52
SCHEMBL1292252 0.80 KMT2A (0.63) NPC1RAB9AKMT2AMEN1RAD52
SCHEMBL13481376 0.80 FGFR1 (0.46) NPC1RAB9AKMT2ARAD52MAPT
SCHEMBL10592001 0.80 HTR7 (0.54) NPC1RAB9AKMT2AMEN1RAD52
SCHEMBL2479803 0.78 CA1 (0.66) NPC1RAB9AKMT2APOLBCACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2050749-B1 PYRIMIDINE DERIVATIVE AS PI3K INHIBITOR AND USE THEREOF CHUGAI PHARMACEUTICAL CO LTD (JP) 2017-11-22 EP disclosed