SCHEMBL19624893

SCHEMBL19624893

Cc1c[nH]c2c(=O)[nH]nc(N)c12

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDPK1 O15530 2/20 0.39
ATAD2 Q6PL18 1/20 0.38
JAK1 P23458 2/20 0.35
TYK2 P29597 2/20 0.35
JAK3 P52333 2/20 0.35
JAK2 O60674 1/20 0.32
LMNA P02545 1/20 0.32
TSHR P16473 1/20 0.32
FGFR1 P11362 1/20 0.30
PRMT5 O14744 1/20 0.30
WDR77 Q9BQA1 1/20 0.30
DYRK1A Q13627 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23815877 0.81 AURKA (0.35) PDPK1JAK2FGFR1DYRK1A
SCHEMBL27188390 0.79 PDPK1 (0.33) PDPK1JAK2FGFR1
SCHEMBL29589071 0.79 PDPK1 (0.43) PDPK1
SCHEMBL25457789 0.73
SCHEMBL19544911 0.72 PDPK1 (0.42) PDPK1JAK1TYK2JAK3JAK2
SCHEMBL11745813 0.67 KDR (0.42) PDPK1JAK1TYK2JAK3JAK2
SCHEMBL22755090 0.66 ATAD2 (0.43) ATAD2
SCHEMBL19533293 0.66 JAK1 (0.36) JAK1TYK2JAK3JAK2LMNA
SCHEMBL8290236 0.64 NOS3 (0.38) LMNA
SCHEMBL24728843 0.64 CHEK1 (0.44) PDPK1FGFR1PRMT5WDR77DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230145305-A1 COMPOUNDS USEFUL AS KINASE INHIBITORS FOCHON BIOSCIENCES, LTD. (CN) 2023-05-11 US disclosed
WO-2021180107-A1 COMPOUNDS USEFUL AS KINASE INHIBITORS FOCHON PHARMACEUTICALS, LTD. (CN) 2021-09-16 WO disclosed
EP-3246317-A1 BTK INHIBITOR Hubei Bio-Pharmaceutical Industrial Technological Institute Inc. (CN) 2017-11-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230145305-A1 COMPOUNDS USEFUL AS KINASE INHIBITORS BTK, ABL1, LCK PDPK1 60/4885ATAD2 2908/4885JAK1 51/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.