SCHEMBL19631558

SCHEMBL19631558

COc1ccc(CN(c2ncns2)S(=O)(=O)c2c(F)cc(N)c(Br)c2F)c(OC)c1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.38
TP53 P04637 1/20 0.35
POLB P06746 2/20 0.33
GAA P10253 1/20 0.32
DHFR P00374 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
HDAC8 Q9BY41 1/20 0.31
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 1/20 0.31
TSHR P16473 1/20 0.31
BMP1 P13497 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19613425 0.92 SCN9A (0.39) SCN9ATP53POLBGAADHFR
SCHEMBL19631626 0.91 SCN9A (0.38) SCN9ATP53POLBGAADHFR
SCHEMBL19631846 0.90 SCN9A (0.38) SCN9ATP53POLBGAADHFR
SCHEMBL22088599 0.88 SCN9A (0.41) SCN9ATP53POLBGAAMEN1
SCHEMBL16011233 0.86 SCN9A (0.41) SCN9ATP53POLBGAAMEN1
SCHEMBL19613979 0.85 SCN9A (0.41) SCN9ATP53POLBGAAMEN1
SCHEMBL21865565 0.85 SCN9A (0.40) SCN9ATP53POLBGAADHFR
SCHEMBL19627736 0.83 SCN9A (0.36) SCN9ABMP1
SCHEMBL28548900 0.83 SCN9A (0.39) SCN9ATP53POLBGAADHFR
SCHEMBL21117665 0.82 SCN9A (0.37) SCN9ATP53POLBGAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10815229-B1 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2020-10-27 US disclosed
US-10662184-B2 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2020-05-26 US disclosed
US-20190194184-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2019-06-27 US disclosed
US-10246453-B2 Benzenesulfonamide compounds and their use as therapeutic agents XENON PHARMACEUTICALS INC. (CA) 2019-04-02 US disclosed
US-20170334902-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2017-11-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-10815229-B1 Benzenesulfonamide compounds and their use as therapeutic agents SCN1A, SCN1B, SCN2B SCN9A 52/4885TP53 1139/4885POLB 3769/4885
US-10246453-B2 Benzenesulfonamide compounds and their use as therapeutic agents SCN1A, SCN1B, SCN2B SCN9A 52/4885TP53 1139/4885POLB 3769/4885
US-20170334902-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN1B, SCN2B SCN9A 52/4885TP53 1139/4885POLB 3769/4885
US-10662184-B2 Benzenesulfonamide compounds and their use as therapeutic agents SCN1A, SCN1B, SCN2B SCN9A 42/4885TP53 1402/4885POLB 3668/4885
US-20190194184-A1 BENZENESULFONAMIDE COMPOUNDS AND THEIR USE AS THERAPEUTIC AGENTS SCN1A, SCN1B, SCN2B SCN9A 42/4885TP53 1402/4885POLB 3668/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.