SCHEMBL19631940

SCHEMBL19631940

C=N/C(=C\C=C/C)C(=O)C1(N2CCN(CCc3ccccc3F)CC2)CCOC(C)(C)C1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 9/20 0.36
SIGMAR1 Q99720 7/20 0.36
KCNH2 Q12809 4/20 0.36
HTR2A P28223 2/20 0.35
OPRD1 P41143 2/20 0.32
OPRK1 P41145 2/20 0.32
CACNA1G O43497 1/20 0.31
ADRA1A P35348 1/20 0.31
HTR2B P41595 1/20 0.31
KMT2A Q03164 2/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
HTR1D P28221 1/20 0.30
HTR1B P28222 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19631885 0.76 HTR2A (0.40) OPRM1SIGMAR1KCNH2HTR2AADRA1A
SCHEMBL19631805 0.72 SIGMAR1 (0.42) OPRM1SIGMAR1KCNH2HTR2ACACNA1G
SCHEMBL19631886 0.71 KCNH2 (0.40) OPRM1SIGMAR1KCNH2HTR2AHTR1D
SCHEMBL19631582 0.68 HTR2A (0.35) OPRM1SIGMAR1KCNH2HTR2A
SCHEMBL19631924 0.67 SLC40A1 (0.35) OPRM1SIGMAR1KCNH2
SCHEMBL19631953 0.67 SIGMAR1 (0.44) OPRM1SIGMAR1KCNH2HTR2A
SCHEMBL19631597 0.67 CYP2A13 (0.48) OPRM1SIGMAR1KCNH2HTR2AHTR1D
SCHEMBL19631945 0.66 SIGMAR1 (0.41) OPRM1SIGMAR1KCNH2HTR2A
SCHEMBL19631920 0.63 SIGMAR1 (0.40) OPRM1SIGMAR1KCNH2KMT2AMEN1
SCHEMBL19631821 0.62 POLB (0.42) OPRM1SIGMAR1KMT2AMEN1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198339-A1 TETRAHYDROPYRAN AND THIOPYRAN DERIVATIVES HAVING MULTIMODAL ACTIVITY AGAINST PAIN LABORATORIOS DEL DR. ESTEVE, S.A. (ES) 2017-11-23 WO disclosed