SCHEMBL19633699

SCHEMBL19633699

COc1cccc(Nc2ccnc3cc(OCc4ccc(OC)c(OC)c4)ccc23)c1

nearest known ligand 0.57

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GAK O14976 6/20 0.57
RIPK2 O43353 2/20 0.57
COQ8A Q8NI60 2/20 0.57
NLK Q9UBE8 2/20 0.57
EGFR P00533 5/20 0.53
HTR1A P08908 2/20 0.49
ADRA1D P25100 2/20 0.49
ADRA1A P35348 2/20 0.49
ADRA1B P35368 2/20 0.49
TGFBR1 P36897 2/20 0.47
KDR P35968 3/20 0.47
RET P07949 1/20 0.47
SRC P12931 1/20 0.47
FERMT2 Q96AC1 1/20 0.46
PDGFRA P16234 1/20 0.45
ABCB1 P08183 1/20 0.45
ERBB3 P21860 1/20 0.45
HTT P42858 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633780 0.91 GAK (0.71) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633519 0.91 GAK (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633565 0.88 MAOB (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633550 0.88 PTK6 (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633676 0.85 GAK (0.68) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633703 0.83 GAK (0.60) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633568 0.81 GAK (0.58) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633513 0.79 GAK (0.56) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633629 0.79 GSK3A (0.61) GAKRIPK2COQ8ANLKEGFR
SCHEMBL30420470 0.79 GAK (0.67) GAKRIPK2COQ8ANLKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed