SCHEMBL19633780

SCHEMBL19633780

COc1cccc(Nc2ccnc3cc(OCc4cc(OC)c(OC)c(OC)c4)ccc23)c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAK O14976 17/20 0.71
RIPK2 O43353 8/20 0.71
COQ8A Q8NI60 8/20 0.71
NLK Q9UBE8 8/20 0.71
EGFR P00533 3/20 0.53
EPHB6 O15197 2/20 0.53
ABL1 P00519 2/20 0.53
ACVR1 Q04771 2/20 0.53
BMPR1B O00238 1/20 0.53
LCK P06239 1/20 0.53
SRC P12931 1/20 0.53
EPHA1 P21709 1/20 0.53
EPHA8 P29322 1/20 0.53
MAP2K5 Q13163 1/20 0.53
HTR1A P08908 2/20 0.50
ADRA1D P25100 2/20 0.50
ADRA1A P35348 2/20 0.50
ADRA1B P35368 2/20 0.50
STK16 O75716 1/20 0.47
AAK1 Q2M2I8 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633699 0.91 GAK (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633519 0.89 GAK (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633550 0.89 PTK6 (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633751 0.88 GAK (0.66) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633565 0.87 MAOB (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633777 0.86 GAK (0.57) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633676 0.86 GAK (0.68) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633703 0.84 GAK (0.60) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633697 0.82 GAK (0.53) GAKRIPK2COQ8ANLKEGFR
SCHEMBL19633778 0.82 GAK (0.69) GAKRIPK2COQ8ANLKEGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed