SCHEMBL19633733

SCHEMBL19633733

C=CCOc1ccc2c(Nc3cccc(F)c3)ccnc2c1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAK O14976 2/20 0.45
ALK Q9UM73 4/20 0.44
TGFBR1 P36897 6/20 0.43
MAPT P10636 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RIPK2 O43353 1/20 0.43
COQ8A Q8NI60 1/20 0.43
NLK Q9UBE8 1/20 0.43
MAP4K4 O95819 1/20 0.43
EGFR P00533 2/20 0.42
FADS1 O60427 1/20 0.42
PKMYT1 Q99640 1/20 0.42
KDR P35968 1/20 0.41
APP P05067 1/20 0.41
NR4A2 P43354 1/20 0.41
RET P07949 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19633513 0.86 GAK (0.56) GAKTGFBR1RIPK2COQ8ANLK
SCHEMBL19633636 0.85 FBP1 (0.51) GAKALKTGFBR1RIPK2COQ8A
SCHEMBL19633548 0.83 GAK (0.48) GAKALKTGFBR1RIPK2COQ8A
SCHEMBL19633632 0.82 GAK (0.62) GAKTGFBR1RIPK2COQ8ANLK
SCHEMBL19633576 0.82 EGFR (0.48) GAKALKTGFBR1RIPK2COQ8A
SCHEMBL19633508 0.82 PTK6 (0.53) GAKALKMAPTEGFRFADS1
SCHEMBL19633621 0.82 KMT2A (0.49) EGFRKDR
SCHEMBL19633572 0.81 GAK (0.46) GAKALKTGFBR1RIPK2COQ8A
SCHEMBL19633640 0.80 GAK (0.60) GAKALKTGFBR1MAP4K4EGFR
SCHEMBL19633566 0.80 SIRT2 (0.47) GAKALKTGFBR1MAP4K4EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198196-A1 QUINOLINE DERIVATIVE HAVING ANTI-TUMOR ACTIVITY 王子厚 2017-11-23 WO disclosed