SCHEMBL19634283

SCHEMBL19634283

COC(=O)c1ccc(C(=O)N(C)CCO)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.55
CYP4A11 Q02928 2/20 0.51
CYP4F2 P78329 1/20 0.50
LMNA P02545 1/20 0.49
MAPT P10636 2/20 0.49
CA1 P00915 2/20 0.48
CA2 P00918 2/20 0.48
TDP1 Q9NUW8 1/20 0.48
CA12 O43570 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
POLB P06746 1/20 0.47
LOXL2 Q9Y4K0 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
HDAC4 P56524 1/20 0.46
TSHR P16473 2/20 0.46
DRD2 P14416 1/20 0.46
HPGD P15428 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10795881 0.87 HDAC4 (0.54) ALDH1A1HDAC4DRD2HPGDSMN1; SMN2
SCHEMBL14640651 0.86 NAMPT (0.49) ALDH1A1LMNAMAPTCA1CA2
SCHEMBL4695349 0.85 NAMPT (0.54) ALDH1A1MAPTCA1CA2TDP1
SCHEMBL23471148 0.84 CYP4F2 (0.55) ALDH1A1CYP4A11CYP4F2MAPTPOLB
SCHEMBL6834844 0.83 DRD2 (0.64) ALDH1A1MAPTCA1CA2MEN1
SCHEMBL28351759 0.82 CA1 (0.52) ALDH1A1CYP4A11LMNAMAPTCA1
SCHEMBL21015888 0.82 HDAC4 (0.46) ALDH1A1CA1CA2CA12CA9
SCHEMBL15768278 0.81 MEN1 (0.57) ALDH1A1LMNAMAPTPOLBMEN1
SCHEMBL13253174 0.81 ALDH1A1 (0.60) ALDH1A1CYP4A11CYP4F2LMNAMAPT
SCHEMBL10076226 0.81 ALDH1A1 (0.50) ALDH1A1MEN1KMT2AHDAC4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed