SCHEMBL19634294

SCHEMBL19634294

COCCN(C)C(=O)c1cccc(CN)c1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LOXL2 Q9Y4K0 4/20 0.56
ATR Q13535 2/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
ROCK2 O75116 1/20 0.46
NAMPT P43490 1/20 0.43
HSD17B1 P14061 1/20 0.42
HSD17B2 P37059 1/20 0.42
ITK Q08881 1/20 0.42
GYS1 P13807 1/20 0.42
LOX P28300 2/20 0.41
PARP1 P09874 1/20 0.41
HDAC4 P56524 1/20 0.40
HTR1A P08908 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
HTR2C P28335 1/20 0.40
SLC7A5 Q01650 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23471221 0.87 MEN1 (0.50) LOXL2ATRMEN1KMT2AROCK2
SCHEMBL23470993 0.86 KMT2A (0.50) LOXL2ATRMEN1KMT2AROCK2
SCHEMBL23471114 0.85 LOXL2 (0.51) LOXL2ATRMEN1KMT2ANAMPT
SCHEMBL18301734 0.85 KMT2A (0.51) ATRMEN1KMT2AROCK2NAMPT
SCHEMBL23471001 0.84 KMT2A (0.47) ATRMEN1KMT2AROCK2NAMPT
SCHEMBL17790195 0.84 ROCK2 (0.51) LOXL2ATRMEN1KMT2AROCK2
SCHEMBL6346088 0.83 ATR (0.51) ATRMEN1KMT2AROCK2NAMPT
SCHEMBL21015933 0.82 KMT2A (0.45) ATRMEN1KMT2AROCK2NAMPT
SCHEMBL12677910 0.81 HPGD (0.54) ATRMEN1KMT2ANAMPTHSD17B2
SCHEMBL21015857 0.81 ROCK2 (0.49) ATRMEN1KMT2AROCK2NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed