SCHEMBL19634412

SCHEMBL19634412

CC(=O)NCc1ccc(C(=O)NCCN2CCN(CC(C)(C)C)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.53
HDAC2 Q92769 2/20 0.53
HDAC8 Q9BY41 1/20 0.53
ALDH1A1 P00352 3/20 0.52
LMNA P02545 2/20 0.52
MAPT P10636 2/20 0.52
SMN1; SMN2 Q16637 2/20 0.52
GAA P10253 1/20 0.52
MAPK1 P28482 1/20 0.52
HTT P42858 1/20 0.52
POLB P06746 2/20 0.50
HDAC1 Q13547 2/20 0.50
NPSR1 Q6W5P4 1/20 0.50
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
NAMPT P43490 2/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR2B P41595 1/20 0.47
HDAC3 O15379 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634461 0.89 HDAC6 (0.55) HDAC6HDAC2HDAC8ALDH1A1LMNA
SCHEMBL19634416 0.88 HDAC6 (0.69) HDAC6HDAC2HDAC8ALDH1A1MAPT
SCHEMBL23471004 0.86 PARP1 (0.48) MAPTPOLBMEN1KMT2ACYP2C9
SCHEMBL19634439 0.86 NPSR1 (0.67) HDAC6HDAC2HDAC8ALDH1A1POLB
SCHEMBL19634686 0.85 HDAC2 (0.55) HDAC6HDAC2HDAC8ALDH1A1LMNA
SCHEMBL19634451 0.85 NPSR1 (0.65) HDAC6HDAC2HDAC8ALDH1A1POLB
SCHEMBL19634402 0.83 KMT2A (0.55) ALDH1A1LMNAMAPTSMN1; SMN2POLB
SCHEMBL23471160 0.83 HASPIN (0.55) HDAC6HDAC2HDAC8ALDH1A1MAPT
SCHEMBL23471332 0.83 HDAC6 (0.52) HDAC6HDAC2HDAC8ALDH1A1MAPT
SCHEMBL19634426 0.83 CD274 (0.67) ALDH1A1POLBNAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed