SCHEMBL19634416

SCHEMBL19634416

CC(=O)NCc1ccc(C(=O)NCCN2CCN(C)CC2)cc1

nearest known ligand 0.69

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.69
HDAC2 Q92769 2/20 0.69
HDAC8 Q9BY41 1/20 0.69
MEN1 O00255 1/20 0.55
KMT2A Q03164 1/20 0.55
HDAC1 Q13547 2/20 0.55
NPSR1 Q6W5P4 1/20 0.54
POLB P06746 3/20 0.53
ALDH1A1 P00352 2/20 0.51
HDAC3 O15379 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2D6 P10635 1/20 0.51
CYP2C9 P11712 1/20 0.51
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
HTR2B P41595 1/20 0.51
NAMPT P43490 1/20 0.51
MAPT P10636 1/20 0.50
RAB9A P51151 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634439 0.91 NPSR1 (0.67) HDAC6HDAC2HDAC8MEN1KMT2A
SCHEMBL19634451 0.90 NPSR1 (0.65) HDAC6HDAC2HDAC8MEN1KMT2A
SCHEMBL19634412 0.88 HDAC6 (0.53) HDAC6HDAC2HDAC8MEN1KMT2A
SCHEMBL23471332 0.87 HDAC6 (0.52) HDAC6HDAC2HDAC8KMT2AHDAC1
SCHEMBL19634426 0.87 CD274 (0.67) POLBALDH1A1NAMPT
SCHEMBL23471160 0.87 HASPIN (0.55) HDAC6HDAC2HDAC8HDAC1NPSR1
SCHEMBL21015348 0.86 HDAC6 (0.64) HDAC6HDAC2HDAC8MEN1KMT2A
SCHEMBL19634745 0.85 PARP1 (0.59) HDAC6HDAC2HDAC8POLBCYP2C9
SCHEMBL11983548 0.82 HDAC2 (0.78) HDAC6HDAC2HDAC8MEN1KMT2A
SCHEMBL23471208 0.82 KMT2A (0.61) HDAC6MEN1KMT2AHDAC1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed