SCHEMBL19634451

SCHEMBL19634451

CC(=O)NCc1ccc(C(=O)NCCN2CCCCC2)cc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.65
CYP1A2 P05177 1/20 0.65
CYP2D6 P10635 1/20 0.65
CYP2C9 P11712 1/20 0.65
POLB P06746 2/20 0.65
NAMPT P43490 2/20 0.61
ALDH1A1 P00352 3/20 0.61
GLA P06280 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58
HPGD P15428 2/20 0.56
KDM4E B2RXH2 1/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
HDAC6 Q9UBN7 2/20 0.55
HDAC1 Q13547 1/20 0.55
CA12 O43570 1/20 0.55
CA9 Q16790 1/20 0.55
HDAC2 Q92769 1/20 0.54
HDAC8 Q9BY41 1/20 0.54
CACNA1G O43497 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634439 0.99 NPSR1 (0.67) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL19634416 0.90 HDAC6 (0.69) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL19634426 0.87 CD274 (0.67) POLBNAMPTALDH1A1HPGDKDM4E
SCHEMBL23471332 0.87 HDAC6 (0.52) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL23471160 0.87 HASPIN (0.55) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL21015947 0.86 NPSR1 (0.61) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL19634412 0.85 HDAC6 (0.53) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL8432036 0.85 NPSR1 (0.70) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL21015946 0.85 NPSR1 (0.62) NPSR1CYP1A2CYP2D6CYP2C9POLB
SCHEMBL10264587 0.83 NPSR1 (0.72) NPSR1CYP1A2CYP2D6CYP2C9POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed