SCHEMBL19634816

SCHEMBL19634816

COCCNC(=O)c1cccc(CNC(C)=O)c1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.57
MMP13 P45452 2/20 0.57
KDM1A O60341 1/20 0.54
HPGD P15428 3/20 0.54
ACACB O00763 1/20 0.53
LMNA P02545 1/20 0.51
CYP3A4 P08684 1/20 0.51
CYP2C9 P11712 1/20 0.51
ROCK1 Q13464 1/20 0.51
MRGPRX4 Q96LA9 1/20 0.51
CHRM2 P08172 1/20 0.50
LOX P28300 1/20 0.48
LOXL2 Q9Y4K0 1/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC10 Q969S8 1/20 0.48
HDAC11 Q96DB2 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634809 0.89 CYP3A4 (0.55) ROCK2MMP13KDM1AHPGDLMNA
SCHEMBL19634811 0.89 ROCK2 (0.50) ROCK2MMP13KDM1AHPGDACACB
SCHEMBL19634574 0.87 KDM1A (0.55) ROCK2MMP13KDM1AHPGDACACB
SCHEMBL19634713 0.86 ROCK2 (0.49) ROCK2MMP13KDM1AHPGDLMNA
SCHEMBL16380331 0.86 ROCK2 (0.53) ROCK2MMP13HPGDLMNACYP3A4
SCHEMBL21015342 0.85 ROCK2 (0.54) ROCK2MMP13KDM1AHPGDLMNA
SCHEMBL23471233 0.84 MRGPRX4 (0.60) ROCK2MMP13KDM1AHPGDACACB
SCHEMBL2056391 0.84 HPGD (0.57) ROCK2KDM1AHPGDACACBMRGPRX4
SCHEMBL8284791 0.84 HPGD (0.57) ROCK2MMP13KDM1AHPGDACACB
SCHEMBL21015600 0.84 MRGPRX4 (0.54) ROCK2MMP13KDM1AHPGDMRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed