SCHEMBL19634574

SCHEMBL19634574

CNCc1cccc(C(=O)NCCOC)c1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.55
ROCK2 O75116 2/20 0.55
HPGD P15428 3/20 0.55
MMP13 P45452 1/20 0.55
MRGPRX4 Q96LA9 1/20 0.52
CHRM2 P08172 1/20 0.51
LOX P28300 2/20 0.49
LOXL2 Q9Y4K0 2/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2C9 P11712 1/20 0.49
ROCK1 Q13464 1/20 0.49
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
LMNA P02545 1/20 0.49
ACACB O00763 1/20 0.48
ALDH1A1 P00352 1/20 0.48
TP53 P04637 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19634816 0.87 ROCK2 (0.57) KDM1AROCK2HPGDMMP13MRGPRX4
SCHEMBL23471211 0.85 ROCK2 (0.51) ROCK2HPGDMMP13MRGPRX4CYP3A4
SCHEMBL8284791 0.85 HPGD (0.57) KDM1AROCK2HPGDMMP13MRGPRX4
SCHEMBL23471233 0.85 MRGPRX4 (0.60) KDM1AROCK2HPGDMMP13MRGPRX4
SCHEMBL2056391 0.85 HPGD (0.57) KDM1AROCK2HPGDMRGPRX4LOX
SCHEMBL21015600 0.85 MRGPRX4 (0.54) KDM1AROCK2HPGDMMP13MRGPRX4
SCHEMBL19634293 0.84 LOXL2 (0.65) KDM1AROCK2HPGDMRGPRX4LOX
SCHEMBL21015342 0.84 ROCK2 (0.54) KDM1AROCK2HPGDMMP13MRGPRX4
SCHEMBL18301728 0.83 HPGD (0.58) KDM1AROCK2HPGDMRGPRX4CHRM2
SCHEMBL17790216 0.82 PARP1 (0.53) ROCK2HPGDMMP13MRGPRX4ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3831841-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T Global Inc. (US) 2021-06-09 EP disclosed
WO-2017200984-A1 NOVEL CYCLOSPORIN DERIVATIVES AND USES THEREOF S&T GLOBAL INC. (US) 2017-11-23 WO disclosed