SCHEMBL19635109

SCHEMBL19635109

OCc1[nH]nc(COCc2ccccc2)c1Br

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.44
CA1 P00915 4/20 0.36
CA2 P00918 2/20 0.36
CA7 P43166 2/20 0.36
CA9 Q16790 2/20 0.36
KDM4E B2RXH2 2/20 0.36
POLB P06746 1/20 0.36
ADORA3 P0DMS8 1/20 0.35
ADORA2A P29274 1/20 0.35
ADORA1 P30542 1/20 0.35
ALDH1A1 P00352 1/20 0.35
PARP1 P09874 3/20 0.33
GRM5 P41594 1/20 0.33
RHEB Q15382 1/20 0.33
GHSR Q92847 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TACR1 P25103 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Benzyl Alcohol SCHEMBL10457557 0.69 TSHR (0.75) TSHRCA1CA2CA7CA9
SCHEMBL19635107 0.69 TSHR (0.42) TSHRKDM4EPOLBALDH1A1RHEB
Hydrogen Peroxide SCHEMBL28758135 0.69 TSHR (0.94) TSHRCA1CA2CA7CA9
SCHEMBL26086950 0.67 TSHR (0.71) TSHRCA1CA2CA7CA9
Ethylene Glycol SCHEMBL130292 0.67 TSHR (0.79) TSHRCA1CA2CA7CA9
SCHEMBL25955862 0.67 TSHR (0.52) TSHRCA1CA2CA7CA9
SCHEMBL21607779 0.67 TSHR (0.47) TSHRGHSRL3MBTL1
SCHEMBL5311581 0.66 TSHR (1.00) TSHRCA1CA2CA7CA9
SCHEMBL27380 0.66 TSHR (1.00) TSHRCA1CA2CA7CA9
Benzene SCHEMBL27997624 0.66 TSHR (1.00) TSHRCA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed