SCHEMBL19635404

SCHEMBL19635404

OCCn1nc(CO)c(Br)c1CN1CCOCC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
KDM4E B2RXH2 2/20 0.40
CSNK2A2 P19784 1/20 0.35
CSNK2B P67870 1/20 0.35
CSNK2A1 P68400 1/20 0.35
CSNK2A3 Q8NEV1 1/20 0.35
CYP2A13 Q16696 1/20 0.34
CYP2C9 P11712 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PIM1 P11309 3/20 0.33
CXCR4 P61073 1/20 0.33
HTT P42858 1/20 0.32
LMNA P02545 2/20 0.32
SLC2A1 P11166 1/20 0.31
GLA P06280 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KMT2A Q03164 2/20 0.30
MEN1 O00255 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19615228 0.87 KMT2A (0.36) ALDH1A1KDM4ECYP2A13ALOX15HTT
SCHEMBL19634925 0.83 LMNA (0.37) ALDH1A1KDM4ECYP2A13CYP2C9ALOX15
SCHEMBL19635653 0.81 PIM1 (0.37) ALDH1A1KDM4EPIM1LMNAGLA
SCHEMBL19635650 0.75 ALDH1A1 (0.37) ALDH1A1KDM4EPIM1LMNAGLA
SCHEMBL19635542 0.74 LMNA (0.40) ALDH1A1KDM4EPIM1LMNAGLA
SCHEMBL19634970 0.74 LMNA (0.37) ALDH1A1KDM4ECYP2A13CYP2C9ALOX15
SCHEMBL19615281 0.69 LMNA (0.39) ALDH1A1KDM4EPIM1LMNASMN1; SMN2
SCHEMBL19616013 0.68 ALDH1A1 (0.38) ALDH1A1KDM4EPIM1LMNAGLA
SCHEMBL19634969 0.64 PARP1 (0.37) ALDH1A1KDM4ECYP2A13CYP2C9ALOX15
SCHEMBL25262333 0.63 KDM4E (0.90) ALDH1A1KDM4EALOX15HSD17B10GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed