SCHEMBL19635446

SCHEMBL19635446

CCOC(=O)c1[nH]nc(CCOC2CCCCO2)c1Br

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
KDM4C Q9H3R0 1/20 0.36
ALDH1A1 P00352 5/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
HSD17B10 Q99714 2/20 0.34
MAPT P10636 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
HPGD P15428 5/20 0.33
GAA P10253 1/20 0.33
TSHR P16473 1/20 0.33
AURKA O14965 1/20 0.32
MAPK10 P53779 1/20 0.32
RIPK1 Q13546 1/20 0.32
DUSP3 P51452 1/20 0.32
MAPK1 P28482 2/20 0.32
HTT P42858 2/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19635900 0.90 ALDH1A1 (0.36) ADORA3MEN1KMT2AALDH1A1NPC1
SCHEMBL29602501 0.78 MEN1 (0.38) ADORA3MEN1KMT2AKDM4CALDH1A1
SCHEMBL19635445 0.78 MEN1 (0.38) ADORA3MEN1KMT2AKDM4CALDH1A1
SCHEMBL14061234 0.77 KDM4C (0.40) ADORA3MEN1KMT2AKDM4CNPC1
SCHEMBL19635447 0.76 KDM4C (0.43) MEN1KMT2AKDM4CNPC1RAB9A
SCHEMBL19635172 0.74 MAPT (0.44) MEN1KMT2AALDH1A1HSD17B10MAPT
SCHEMBL19635441 0.74 MAPT (0.44) MEN1KMT2AALDH1A1HSD17B10MAPT
SCHEMBL1809242 0.72 NPC1 (0.42) ADORA3MEN1KMT2AKDM4CALDH1A1
SCHEMBL24524644 0.72 MEN1 (0.38) ADORA3MEN1KMT2AALDH1A1NPC1
SCHEMBL19635605 0.71 ALDH1A1 (0.43) KMT2AALDH1A1RAB9AHSD17B10L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3458459-B1 MACROCYCLIC INDOLE DERIVATIVES BAYER AG (DE) 2022-04-27 EP disclosed
WO-2017198341-A1 MACROCYCLIC INDOLE DERIVATIVES BAYER AKTIENGESELLSCHAFT (DE) 2017-11-23 WO disclosed