SCHEMBL19635796

SCHEMBL19635796

CC#CC(=O)N1CCC[C@@H](n2nc(-c3ccc(Oc4ccc(Cl)cn4)cc3)c3c(N)ncnc32)C1

nearest known ligand 0.77

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BTK Q06187 20/20 0.77
ITK Q08881 2/20 0.77
EGFR P00533 1/20 0.77
LCK P06239 1/20 0.77
BLK P51451 2/20 0.62
FGR P09769 1/20 0.61
FLT3 P36888 1/20 0.61
CSK P41240 1/20 0.61
JAK3 P52333 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21330631 0.90 BTK (0.91) BTKITKEGFRLCKBLK
SCHEMBL21330635 0.90 BTK (0.91) BTKITKEGFRLCKBLK
SCHEMBL28370674 0.90 BTK (0.76) BTKITKEGFRLCKBLK
SCHEMBL28370673 0.90 BTK (0.76) BTKITKEGFRLCKBLK
SCHEMBL410333 0.87 BTK (1.00) BTKITKEGFRLCKBLK
SCHEMBL29663941 0.87 BTK (1.00) BTKITKEGFRLCKBLK
SCHEMBL443936 0.87 BTK (1.00) BTKITKEGFRLCKBLK
SCHEMBL19635192 0.87 BTK (0.64) BTKITKEGFRLCKBLK
SCHEMBL19635202 0.87 BTK (0.64) BTKITKEGFRLCKBLK
SCHEMBL19635227 0.87 BTK (0.64) BTKITKEGFRLCKBLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017198049-A1 PYRAZOLOPYRIMIDINE DERIVATIVE AS BTK INHIBITOR AND PREPARATION METHOD AND PHARMACEUTICAL COMPOSITION THEREOF 浙江予川医药科技有限公司 2017-11-23 WO disclosed