SCHEMBL19636447

SCHEMBL19636447

C=C1C(=C)[C@H](N(Cc2ccccc2)S(C)(=O)=O)[C@H]1N(Cc1ccccc1)S(C)(=O)=O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.44
ALDH1A1 P00352 3/20 0.43
POLB P06746 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CA2 P00918 1/20 0.42
TSHR P16473 2/20 0.40
SLC6A2 P23975 3/20 0.39
SLC6A4 P31645 3/20 0.39
KCNH2 Q12809 3/20 0.39
SLC6A3 Q01959 2/20 0.39
NR3C2 P08235 1/20 0.39
DPP4 P27487 1/20 0.39
DPP9 Q86TI2 1/20 0.39
DPP7 Q9UHL4 1/20 0.39
PER2 O15055 1/20 0.38
CRY1 Q16526 1/20 0.38
CRY2 Q49AN0 1/20 0.38
MCHR1 Q99705 1/20 0.37
AOC3 Q16853 1/20 0.37
NR3C1 P04150 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19636592 0.79 CNR2 (0.55) ALDH1A1POLBTSHRMCHR1NR3C1
SCHEMBL2492170 0.71 TSHR (0.53) ALDH1A1POLBSMN1; SMN2CA2TSHR
SCHEMBL10312253 0.71 ALDH1A1 (0.64) ALDH1A1POLBSMN1; SMN2CA2TSHR
SCHEMBL2057187 0.70 ALDH1A1 (0.54) ALDH1A1POLBSMN1; SMN2CA2TSHR
SCHEMBL27410092 0.69 ALDH1A1 (0.49) ALDH1A1POLBSMN1; SMN2CA2TSHR
SCHEMBL20679705 0.68 ALDH1A1 (0.45) ALDH1A1POLBSMN1; SMN2CA2TSHR
SCHEMBL24571678 0.67 TSHR (0.68) ALDH1A1POLBSMN1; SMN2CA2TSHR
SCHEMBL12808838 0.67 ALDH1A1 (0.60) ALDH1A1POLBSMN1; SMN2TSHRMEN1
SCHEMBL13306986 0.67 ALDH1A1 (0.50) ALDH1A1POLBSMN1; SMN2CA2TSHR
SCHEMBL2103432 0.67 SMN1; SMN2 (0.58) ALDH1A1POLBSMN1; SMN2CA2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107400036-B A method of synthesis 1,2- dimethylene cyclobutane chipal compounds 中国科学院福建物质结构研究所 2019-09-20 CN disclosed
CN-107400036-A A kind of method of synthesis 1,2- dimethylene cyclobutane chipal compounds 中国科学院福建物质结构研究所 2017-11-28 CN disclosed
WO-2017197670-A1 METHOD FOR SYNTHESIZING 1,2-DIMETHYLENE CYCLOBUTANE CHIRAL COMPOUND 中国科学院福建物质结构研究所 2017-11-23 WO disclosed