SCHEMBL1963739

SCHEMBL1963739

NNc1[c]cccn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL933811 0.76
SCHEMBL28149711 0.71
SCHEMBL6015000 0.71 IDO1 (0.34)
SCHEMBL1385358 0.71
SCHEMBL12470502 0.71 KDM4E (0.44)
SCHEMBL8725876 0.70 HSD17B10 (0.42)
SCHEMBL8922325 0.69 CYP2C19 (0.51)
SCHEMBL6647364 0.69 MEN1 (0.44)
SCHEMBL5386852 0.69 GLO1 (0.41)
SCHEMBL2066722 0.69 KDM4E (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9175036-B2 Antimicrobial water treatment membranes and production thereof BEN-GURION UNVERSITY OF THE NEGEV RESEARCH AND DEVELOPMENT AUTHORITY (IL) 2015-11-03 US disclosed
US-20140238939-A1 IMMOBILIZATION OF ANTIMICROBIAL POLYMERS ON RO MEMBRANE TO REDUCE BIOFILM GROWTH AND BIOFOULING WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2014-08-28 US disclosed
US-20120325748-A1 ANTIMICROBIAL WATER TREATMENT MEMBRANES AND PRODUCTION THEREOF BAR-ILAN UNIVERSITY (IL) 2012-12-27 US disclosed
WO-2012172547-A1 IMMOBILIZATION OF ANTIMICROBIAL POLYMERS ON RO MEMBRANE TO REDUCE BIOFILM GROWTH AND BIOFOULING BEN-GURION UNIVERSITY OF THE NEGEV RESEARCH AND DEVELOPMENT AUTHORITY (IL) 2012-12-20 WO disclosed
EP-2509614-A1 ANTIMICROBIAL WATER TREATMENT MEMBRANES AND PRODUCTION THEREOF Ben-Gurion University Of The Negev Research And Development Authority (IL) 2012-10-17 EP disclosed
US-20120121641-A1 MHC OLIGOMER AND METHOD OF MAKING THE SAME PROIMMUNE LIMITED (GB) 2012-05-17 US disclosed
EP-1844072-B1 MHC OLIGOMER AND METHOD OF MAKING THE SAME PROIMMUNE LTD (GB) 2012-04-04 EP disclosed
WO-2011070573-A1 ANTIMICROBIAL WATER TREATMENT MEMBRANES AND PRODUCTION THEREOF BEN-GURION UNIVERSITY OF THE NEGEV RESEARCH AND DEVELOPMENT AUTHORITY (IL) 2011-06-16 WO disclosed
US-20100012880-A1 MAGNETIC PARTICLES AND METHODS OF MAKING AND USING THE SAME COLUMBUS NANOWORKS, INC. (US) 2010-01-21 US disclosed
EP-2062271-A2 MAGNETIC PARTICLES AND METHODS OF MAKING AND USING THE SAME Columbus Nanoworks, Inc. (US) 2009-05-27 EP disclosed
US-20080207485-A1 Mhc Oligomer And Method Of Making The Same PROIMMUNE LIMITED 2008-08-28 US disclosed
WO-2008030862-A2 MAGNETIC PARTICLES AND METHODS OF MAKING AND USING THE SAME COLUMBUS NANOWORKS, INC. (US) 2008-03-13 WO disclosed
CN-101111520-A MHC oligomers and methods for making same PROIMMUNE LTD (GB) 2008-01-23 CN disclosed
US-20070258969-A1 Compositions and methods for targeting metastatic tumors using multivalent ligand-linked carbohydrate polymers GALECTIN THERAPEUTICS, INC. 2007-11-08 US disclosed
EP-1844072-A1 MHC OLIGOMER AND METHOD OF MAKING THE SAME ProImmune Limited (GB) 2007-10-17 EP disclosed
EP-1734819-A1 COMPOSITIONS AND METHODS FOR TARGETING METASTATIC TUMORS USING MULTIVALENT LIGAND-LINKED CARBOHYDRATE POLYMERS Pro-Pharmaceuticals, Inc. (US) 2006-12-27 EP disclosed
WO-2006082387-A1 MHC OLIGOMER AND METHOD OF MAKING THE SAME PROIMMUNE LIMITED (GB) 2006-08-10 WO disclosed
US-20060008907-A1 Control of gene expression via light activated RNA interference THE CURATORS OF THE UNIVERSITY OF MISSOURI 2006-01-12 US disclosed
WO-2005092097-A1 COMPOSITIONS AND METHODS FOR TARGETING METASTATIC TUMORS USING MULTIVALENT LIGAND-LINKED CARBOHYDRATE POLYMERS PRO-PHARMACEUTICALS, INC. (US) 2005-10-06 WO disclosed