SCHEMBL1963928

SCHEMBL1963928

O[C@H]1CCN(Cc2ccccc2)C[C@@H]1F

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.58
FUCA1 P04066 2/20 0.56
SLC18A3 Q16572 4/20 0.53
ACHE P22303 2/20 0.51
BCHE P06276 1/20 0.51
BACE1 P56817 1/20 0.51
SIGMAR1 Q99720 2/20 0.51
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C19 P33261 1/20 0.50
GBA1 P04062 1/20 0.50
CCR3 P51677 1/20 0.50
GRIN1 Q05586 1/20 0.49
GRIN2B Q13224 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30195485 1.00 ALDH1A1 (0.58) ALDH1A1FUCA1SLC18A3ACHEBCHE
SCHEMBL5157969 0.85 FUCA1 (0.66) ALDH1A1FUCA1SLC18A3ACHEBCHE
SCHEMBL5157349 0.85 FUCA1 (0.66) ALDH1A1FUCA1SLC18A3ACHEBCHE
SCHEMBL30014513 0.85 FUCA1 (0.71) ALDH1A1FUCA1SLC18A3SIGMAR1GBA1
SCHEMBL20484873 0.84 HTR2A (0.48) ALDH1A1SLC18A3SIGMAR1CYP1A2CYP3A4
SCHEMBL20484874 0.84 HTR2A (0.48) ALDH1A1SLC18A3SIGMAR1CYP1A2CYP3A4
SCHEMBL20485039 0.84 HTR2A (0.48) ALDH1A1SLC18A3SIGMAR1CYP1A2CYP3A4
SCHEMBL4436419 0.83 ACHE (0.58) ACHESIGMAR1
SCHEMBL14211659 0.81 GBA1 (0.52) ALDH1A1FUCA1ACHEBCHEBACE1
SCHEMBL29927577 0.81 GBA1 (0.52) ALDH1A1FUCA1ACHEBCHEBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2334677-A1 TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS Array Biopharma, Inc. (US) 2011-06-22 EP disclosed
WO-2010022076-A1 TRIAZOLOPYRIDINE COMPOUNDS AS PIM KINASE INHIBITORS ARRAY BIOPHARMA INC. (US) 2010-02-25 WO disclosed